Compile Data Set for Download or QSAR
Found 191 with Last Name = 'nishida' and Initial = 'a'
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi:  0.0680nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.0970nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)copy SMILEScopy InChI
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))copy SMILEScopy InChI
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM82403(CAS_108186 | CI-988 | NSC_108186)copy SMILEScopy InChI
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)copy SMILEScopy InChI
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)copy SMILEScopy InChI
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM82480(YM022 S-isomer)copy SMILEScopy InChI
Affinity DataKi:  140nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi:  260nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM82480(YM022 S-isomer)copy SMILEScopy InChI
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50061220(1-((S)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)copy SMILEScopy InChI
Affinity DataKi:  5.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM82403(CAS_108186 | CI-988 | NSC_108186)copy SMILEScopy InChI
Affinity DataKi:  6.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetD(1A) dopamine receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetAlpha-2C adrenergic receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGlutamate receptor 3(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3Z2FPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50286892(1-[(R)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99553
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056102((R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50286884(1-{1-[2-(1-Methyl-cyclopentyl)-2-oxo-ethyl]-2-oxo-...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99553
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Ability to displace [125I]-CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99553
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8DGT
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056103(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056093(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056099(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056101(1-[(R)-2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-phenyl-2,...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50286903(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8DGT
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50286897(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-2-yl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.130nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]-CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8DGT
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056092(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.140nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056091(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3...)copy SMILEScopy InChI
Affinity DataIC50: 0.160nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056089(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056095(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Yamanouchi Pharmaceutical Co. Ltd.

Curated by PDSP Ki Database
LigandPNGBDBM50056098(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMAssay Description:Inhibitory concentration against radioligand [125I]-CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4BBQPubMed
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