Compile Data Set for Download or QSAR
Found 127 with Last Name = 'orzeszko' and Initial = 'a'
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34046(iodinated benzimidazole, 9a)copy SMILEScopy InChI
Affinity DataKi:  19nM ΔG°:  -45.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  23nM ΔG°:  -45.4kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34044(iodinated benzimidazole, 7a)copy SMILEScopy InChI
Affinity DataKi:  24nM ΔG°:  -45.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359842(CHEMBL1928905)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34051(iodinated benzimidazole, 14)copy SMILEScopy InChI
Affinity DataKi:  27nM ΔG°:  -44.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  37nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34054(iodinated benzimidazole, 17)copy SMILEScopy InChI
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34052(iodinated benzimidazole, 15)copy SMILEScopy InChI
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  54nM ΔG°:  -43.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34055(iodinated benzimidazole, 21)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34048(iodinated benzimidazole, 11a)copy SMILEScopy InChI
Affinity DataKi:  70nM ΔG°:  -42.5kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34043(iodinated benzimidazole, 6a)copy SMILEScopy InChI
Affinity DataKi:  75nM ΔG°:  -42.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)copy SMILEScopy InChI
Affinity DataKi:  77nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359844(CHEMBL1928907)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  83nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359846(CHEMBL1233807)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359844(CHEMBL1928907)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359841(CHEMBL1928904)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34050(iodinated benzimidazole, 13a)copy SMILEScopy InChI
Affinity DataKi:  90nM ΔG°:  -41.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359847(CHEMBL1928909)copy SMILEScopy InChI
Affinity DataKi:  93nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  97nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34040(iodinated benzimidazole, 3a)copy SMILEScopy InChI
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156673(((4,5,6,7-tetrabromo-1H-benzimidazol-2-yl)sulfanyl...)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156680(2-(dimethylamino)-1-methyl-4,5,6,7-tetrabromo-1Hbe...)copy SMILEScopy InChI
Affinity DataKi:  109nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM34053(iodinated benzimidazole, 16)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  112nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359840(CHEMBL1928903)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into P2B substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34047(iodinated benzimidazole, 10a)copy SMILEScopy InChI
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34049(iodinated benzimidazole, 12a)copy SMILEScopy InChI
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34056(iodinated benzimidazole, 23)copy SMILEScopy InChI
Affinity DataKi:  130nM ΔG°:  -40.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ860PPubMed
TargetCasein kinase II subunit alpha'(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  133nMAssay Description:Inhibition of human CK2 alpha' catalytic subunit expressed in Escherichia coli BE21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50359843(CHEMBL1928906)copy SMILEScopy InChI
Affinity DataKi:  137nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
The John Paul II Catholic University of Lublin

Curated by ChEMBL
LigandPNGBDBM50156670(2-(dimethylamino)-4,5,6,7-tetrabromo-1H-benzimidaz...)copy SMILEScopy InChI
Affinity DataKi:  139nMAssay Description:Inhibition of human CK2 alpha catalytic subunit expressed in Escherichia coli BL21 (DE3) assessed as [33P]gamma-ATP incorporation into RRRADDSDDDDD s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377944PubMed
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