Compile Data Set for Download or QSAR
Found 61 with Last Name = 'ozawa' and Initial = 'a'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246834(CHEMBL4067640)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246823(CHEMBL4071277)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246826(CHEMBL4084577)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246835(CHEMBL4077474)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246819(CHEMBL4073220)copy SMILEScopy InChI
Affinity DataKi:  58nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246827(CHEMBL4100236)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246823(CHEMBL4071277)copy SMILEScopy InChI
Affinity DataKi:  85nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246834(CHEMBL4067640)copy SMILEScopy InChI
Affinity DataKi:  125nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246826(CHEMBL4084577)copy SMILEScopy InChI
Affinity DataKi:  167nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246823(CHEMBL4071277)copy SMILEScopy InChI
Affinity DataKi:  184nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246831(CHEMBL4089792)copy SMILEScopy InChI
Affinity DataKi:  221nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246835(CHEMBL4077474)copy SMILEScopy InChI
Affinity DataKi:  281nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246843(CHEMBL4092784)copy SMILEScopy InChI
Affinity DataKi:  314nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246830(CHEMBL4061680)copy SMILEScopy InChI
Affinity DataKi:  321nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246825(CHEMBL4068559)copy SMILEScopy InChI
Affinity DataKi:  325nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246832(CHEMBL4070832)copy SMILEScopy InChI
Affinity DataKi:  361nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246825(CHEMBL4068559)copy SMILEScopy InChI
Affinity DataKi:  361nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246822(CHEMBL4098322)copy SMILEScopy InChI
Affinity DataKi:  448nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246827(CHEMBL4100236)copy SMILEScopy InChI
Affinity DataKi:  471nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246839(CHEMBL4070343)copy SMILEScopy InChI
Affinity DataKi:  474nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246820(CHEMBL4100067)copy SMILEScopy InChI
Affinity DataKi:  577nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246843(CHEMBL4092784)copy SMILEScopy InChI
Affinity DataKi:  601nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246832(CHEMBL4070832)copy SMILEScopy InChI
Affinity DataKi:  628nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246831(CHEMBL4089792)copy SMILEScopy InChI
Affinity DataKi:  633nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246833(CHEMBL4088860)copy SMILEScopy InChI
Affinity DataKi:  640nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246819(CHEMBL4073220)copy SMILEScopy InChI
Affinity DataKi:  644nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246824(CHEMBL4081815)copy SMILEScopy InChI
Affinity DataKi:  652nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246838(CHEMBL4097518)copy SMILEScopy InChI
Affinity DataKi:  704nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246842(CHEMBL4059898)copy SMILEScopy InChI
Affinity DataKi:  711nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246826(CHEMBL4084577)copy SMILEScopy InChI
Affinity DataKi:  716nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246836(CHEMBL4102525)copy SMILEScopy InChI
Affinity DataKi:  771nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246828(CHEMBL4074282)copy SMILEScopy InChI
Affinity DataKi:  863nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-5/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246823(CHEMBL4071277)copy SMILEScopy InChI
Affinity DataKi:  957nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4alpha5 nAChR expressed in HEK cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246823(CHEMBL4071277)copy SMILEScopy InChI
Affinity DataKi:  964nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246826(CHEMBL4084577)copy SMILEScopy InChI
Affinity DataKi:  1.03E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246830(CHEMBL4061680)copy SMILEScopy InChI
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246833(CHEMBL4088860)copy SMILEScopy InChI
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246842(CHEMBL4059898)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246844(CHEMBL4089684)copy SMILEScopy InChI
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246841(CHEMBL4090594)copy SMILEScopy InChI
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246821(CHEMBL4062628)copy SMILEScopy InChI
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-5/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246826(CHEMBL4084577)copy SMILEScopy InChI
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4alpha5 nAChR expressed in HEK cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246840(CHEMBL4097405)copy SMILEScopy InChI
Affinity DataKi:  2.25E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246829(CHEMBL70624)copy SMILEScopy InChI
Affinity DataKi:  3.75E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246837(CHEMBL4094784)copy SMILEScopy InChI
Affinity DataKi:  4.96E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246836(CHEMBL4102525)copy SMILEScopy InChI
Affinity DataKi:  1.23E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246828(CHEMBL4074282)copy SMILEScopy InChI
Affinity DataKi:  1.81E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246837(CHEMBL4094784)copy SMILEScopy InChI
Affinity DataKi:  1.87E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246841(CHEMBL4090594)copy SMILEScopy InChI
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246820(CHEMBL4100067)copy SMILEScopy InChI
Affinity DataKi:  2.45E+4nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1V5MPubMed
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