TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena
Curated by ChEMBL
2-Universit£ di Siena
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena
Curated by ChEMBL
2-Universit£ di Siena
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutantMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027](Human immunodeficiency virus type 1 group M subtyp...)
Universita di Siena
Universita di Siena
Affinity DataKi: 30nM ΔG°: -44.7kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of the RNA-dependent DNA polymerase activity of the HIV-1 reverse transcriptase enzyme was measured using a primer extension assay. Th...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena
Curated by ChEMBL
2-Universit£ di Siena
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena
Curated by ChEMBL
2-Universit£ di Siena
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027,V694A]/[588-1147,V694A](Human immunodeficiency virus type 1)
Universita di Siena
Universita di Siena
Affinity DataKi: 40nMAssay Description:The inhibition of the RNA-dependent DNA polymerase activity of the HIV-1 reverse transcriptase enzyme was measured using a primer extension assay. Th...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena
Curated by ChEMBL
2-Universit£ di Siena
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena
Curated by ChEMBL
2-Universit£ di Siena
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena
Curated by ChEMBL
2-Universit£ di Siena
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of HIV1 free wild type reverse transcriptaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase/poly(rA)/oligo(dT) DNA binary complexMore data for this Ligand-Target Pair