Compile Data Set for Download or QSAR
Found 475 with Last Name = 'samuele' and Initial = 'a'
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477178(CHEMBL239063)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM2325(2-(cyclopentylsulfanyl)-6-[1-(2,6-difluorophenyl)e...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477201(CHEMBL394990)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477199(CHEMBL239342)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477179(CHEMBL399016)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477179(CHEMBL399016)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50339536((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319ZQ9PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena

Curated by ChEMBL
LigandPNGBDBM50339536((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319ZQ9PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477199(CHEMBL239342)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477188(CHEMBL239337)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477198(CHEMBL239064)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477188(CHEMBL239337)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477200(CHEMBL396816)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477200(CHEMBL396816)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477185(CHEMBL239338)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477196(CHEMBL393696)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena

Curated by ChEMBL
LigandPNGBDBM2325(2-(cyclopentylsulfanyl)-6-[1-(2,6-difluorophenyl)e...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetGag-Pol polyprotein [588-1027](Human immunodeficiency virus type 1 group M subtyp...)
Universita di Siena

LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  30nM ΔG°:  -44.7kJ/molepH: 7.5 T: 2°CAssay Description:The inhibition of the RNA-dependent DNA polymerase activity of the HIV-1 reverse transcriptase enzyme was measured using a primer extension assay. Th...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477186(CHEMBL238907)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase V179D mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena

Curated by ChEMBL
LigandPNGBDBM50339522((+/-)-6-Ethyl-6-[4-[(4-bromophenylthio)methyl]phen...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase L100I mutant/poly(rA)/oligo(dT) DNA/dTTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319ZQ9PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477198(CHEMBL239064)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477189(CHEMBL239281)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477189(CHEMBL239281)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetGag-Pol polyprotein [588-1027,V694A]/[588-1147,V694A](Human immunodeficiency virus type 1)
Universita di Siena

LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:The inhibition of the RNA-dependent DNA polymerase activity of the HIV-1 reverse transcriptase enzyme was measured using a primer extension assay. Th...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477188(CHEMBL239337)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477185(CHEMBL239338)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477186(CHEMBL238907)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477179(CHEMBL399016)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477180(CHEMBL238701)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477186(CHEMBL238907)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477198(CHEMBL239064)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2JXBPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477199(CHEMBL239342)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477197(CHEMBL391164)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of wild type HIV1 3B reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
2-Universit£ di Siena

Curated by ChEMBL
LigandPNGBDBM50477185(CHEMBL239338)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of HIV1 reverse transcriptase K103N mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50477195(CHEMBL239120)copy SMILEScopy InChI
Affinity DataKi:  90nMAssay Description:Inhibition of HIV1 reverse transcriptase V106A mutantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H99803PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50339536((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...)copy SMILEScopy InChI
Affinity DataKi:  90nMAssay Description:Inhibition of HIV1 free wild type reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319ZQ9PubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ degli Studi di Roma La Sapienza

Curated by ChEMBL
LigandPNGBDBM50339536((+/-)-6-Ethyl-6-[4-[(2-chloro-4-fluorophenylthio)m...)copy SMILEScopy InChI
Affinity DataKi:  90nMAssay Description:Inhibition of HIV1 wild type reverse transcriptase/poly(rA)/oligo(dT) DNA binary complexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319ZQ9PubMed
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