Compile Data Set for Download or QSAR
Found 1021 with Last Name = 'scholz' and Initial = 'a'
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180827(US9133171, 32)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
LigandPNGBDBM259295(US9499547, 36)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2736PVKUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM187124(US9670161, 5 N-{6-(Difluoromethyl)-4-[(methylsulfo...)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 8.0Assay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29G5K05US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333401(2-{[3-(Furo[2,3-c]pyridin-2-yl)imidazo[1,2-b]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333402(2-{[3-(Furo[3,2-c]pyridin-2-yl)imidazo[1,2-b]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bayer HealthCare AG

Curated by ChEMBL
LigandPNGBDBM50134989(CHEMBL3746640)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of MEK1 in human HeLa-MaTu matched pair cells assessed as reduction in ERK phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38NNPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180836(US9133171, 41)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180837(US9133171, 42)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180843(US9133171, 48)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180815(US9133171, 20)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180819(US9133171, 24)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180824(US9133171, 29 | US9133171, 30 | US9133171, 31)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180799(US9133171, 13 | US9133171, 14 | US9133171, 4)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180823(US9133171, 28)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180824(US9133171, 29 | US9133171, 30 | US9133171, 31)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180824(US9133171, 29 | US9133171, 30 | US9133171, 31)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180851(US9133171, 56)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180853(US9133171, 58)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetIsoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D](Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM223024(US9320737, II.1)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:For the assay 50 mL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2F00US Patent
TargetIsoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D](Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM223030(US9320737, III.3)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:For the assay 50 mL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2F00US Patent
TargetIsoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) 344D](Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM223043(US9320737, IV.2)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:For the assay 50 mL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22V2F00US Patent
LigandPNGBDBM259295(US9499547, 36)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:MKNK1-inhibitory activity at high ATP of compounds of the present invention after their preincubation with MKNK1 was quantified employing the TR-FRET...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2736PVKUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM170515(US9669034, 90 (rac)-4-{4-Fluoro-2-[(3-fluorobenzyl...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22Z13PGUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM175041(US9669034, 99 (rac)-4-{4-Fluoro-2-[(2-methylprop-2...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22Z13PGUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM176781(US9669034, 104 (rac)-4-{4-Fluoro-2-[(3,4,5-trifluo...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22Z13PGUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM179848(US9669034, 113 (rac)-[Cyclopropyl(3-{[4-(4-fluoro-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22Z13PGUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM187120(US9670161, 1 5-Fluoro-4-(4-fluoro-2-methoxyphenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0Assay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29G5K05US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM187120(US9670161, 1 5-Fluoro-4-(4-fluoro-2-methoxyphenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0Assay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29G5K05US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM170016(US9669034, 82 (rac)-4-{4-Fluoro-2-[(2-fluoropyridi...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0 T: 2°CAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22Z13PGUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM187121(US9670161, 2 5-Fluoro-4-(4-fluoro-2-methoxyphenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0Assay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29G5K05US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM187122(US9670161, 3 5-Fluoro-4-(4-fluoro-2-methoxyphenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0Assay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29G5K05US Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM187124(US9670161, 5 N-{6-(Difluoromethyl)-4-[(methylsulfo...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 8.0Assay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29G5K05US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333382(3-[(1R)-1-{[3-(1- Benzofuran-2- yl)imidazo[1,2-b]p...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333390(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180828(US9133171, 33 | US9133171, 34 | US9133171, 35)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180853(US9133171, 58)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180856(US9133171, 61 | US9133171, 62 | US9133171, 63)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180859(US9133171, 64)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180812(US9133171, 17 | US9133171, 18 | US9133171, 19)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180824(US9133171, 29 | US9133171, 30 | US9133171, 31)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchased fro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180819(US9133171, 24)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180824(US9133171, 29 | US9133171, 30 | US9133171, 31)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180836(US9133171, 41)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180856(US9133171, 61 | US9133171, 62 | US9133171, 63)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM180859(US9133171, 64)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were purchase from...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SX6C0WUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM168387(US9669034, 6 (rac)-4-[2-(Benzyloxy)-4-fluorophenyl...)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q22Z13PGUS Patent
LigandPNGBDBM259297(US9499547, 38)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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BindingDB Entry DOI: 10.7270/Q2736PVKUS Patent
LigandPNGBDBM259298(US9499547, 39)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2736PVKUS Patent
LigandPNGBDBM259260(US9499547, 1)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2736PVKUS Patent
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM258868(US9499492, 20)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 8.0 T: 2°CAssay Description:Method 1a: Recombinant full-length His-tagged human CDK9 and CycT1, expressed in insect cells and purified by Ni-NTA affinity chromatography, were pu...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q2GH9GW0US Patent
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