Compile Data Set for Download or QSAR
Found 74 with Last Name = 'varnek' and Initial = 'a'
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50004058((2S)-2-(butylsulfonylamino)-3-[4-(4-piperidin-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354350(CHEMBL1836344)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354350(CHEMBL1836344)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124560(CHEMBL3623706)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity against integrin alpha2bbeta3 open form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354352(CHEMBL1836347)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354355(CHEMBL1836351)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354352(CHEMBL1836347)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354355(CHEMBL1836351)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354351(CHEMBL1836345)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354351(CHEMBL1836345)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124522(CHEMBL3623709)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity against integrin alpha2bbeta3 closed form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354356(CHEMBL1836355)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50078448(3-{[3-Oxo-2-(2-piperidin-4-yl-ethyl)-2,3-dihydro-1...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Antagonist activity at integrin alpha2beta3-mediated aggregation in ADP-stimulated human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124559(CHEMBL3623707)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Antagonist activity against integrin alpha2bbeta3 open form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50004058((2S)-2-(butylsulfonylamino)-3-[4-(4-piperidin-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Antagonist activity against integrin alpha2bbeta3 closed form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregatio...More data for this Ligand-Target Pair
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50004058((2S)-2-(butylsulfonylamino)-3-[4-(4-piperidin-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Antagonist activity against integrin alpha2bbeta3 open form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregationMore data for this Ligand-Target Pair
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354354(CHEMBL1836350)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354354(CHEMBL1836350)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124573(CHEMBL1472460)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Antagonist activity against integrin alpha2bbeta3 in human platelet rich plasmaMore data for this Ligand-Target Pair
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124510(CHEMBL3623710)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity against integrin alpha2bbeta3 closed form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124558(CHEMBL3623708)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Antagonist activity against integrin alpha2bbeta3 closed form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465543(CHEMBL4278778)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465543(CHEMBL4278778)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354348(CHEMBL1836342)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354348(CHEMBL1836342)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465544(CHEMBL4285802)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124571(CHEMBL3623501)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Antagonist activity against integrin alpha2bbeta3 open form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354353(CHEMBL1836348)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354353(CHEMBL1836348)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465540(CHEMBL4282396)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465534(CHEMBL4288560)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465539(CHEMBL4292433)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465536(CHEMBL4282793)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465541(CHEMBL4284735)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465537(CHEMBL4286225)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465533(CHEMBL4289190)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465535(CHEMBL4278314)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50124561(CHEMBL3621231)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Antagonist activity against integrin alpha2bbeta3 open form in human platelet rich plasma assessed as inhibition of ADP-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465545(CHEMBL4293000)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465546(CHEMBL4277865)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465538(CHEMBL4284197)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354349(CHEMBL1836343)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of FITC-labeled fibrinogen from alpha2beta3 in human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1XNSPubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50354349(CHEMBL1836343)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of FITC-labeled fibrinogen binding to integrin alpha2bbeta3 receptor in human platelets by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81FGXPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465548(CHEMBL4286686)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465547(CHEMBL4292615)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465542(CHEMBL4281327)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465551(CHEMBL4290684)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50536995(CHEMBL4572971)copy SMILEScopy InChI
Affinity DataIC50: 8.81E+3nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TZDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50536988(CHEMBL4570691)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of BRD4 (unknown origin) measured after 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TZDPubMed
TargetIntegrin alpha-2/beta-3(Homo sapiens (Human))
A.V. Bogatsky Physico-Chemical Institute of the National Academy of Sciences of Ukraine

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)copy SMILEScopy InChI
Affinity DataIC50: 1.25E+4nMAssay Description:Antagonist activity against integrin alpha2bbeta3 in human platelet rich plasmaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN68MBPubMed
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