Compile Data Set for Download or QSAR
Found 279 with Last Name = 'vilas-zornoza' and Initial = 'a'
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50105327(JNJ-26481585 | Quisinostat)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Inhibition of recombinant full length C-terminal FLAG His-tagged human HDAC1 expressed in baculovirus infected Sf21 insect cells using RHK-K(Ac)-AMC ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50105327(JNJ-26481585 | Quisinostat)copy SMILEScopy InChI
Affinity DataIC50: 0.330nMAssay Description:Inhibition of recombinant full length C-terminal GST fusion-tagged human HDAC2 expressed in baculovirus infected insect cells using RHK-K(Ac)-AMC as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281305(CHEMBL4162206)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Non-competitive inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of 2 to 640 uM SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281300(CHEMBL4170225)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281305(CHEMBL4162206)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281305(CHEMBL4162206)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Competitive inhibition of human G9a using 40 to 2560 nM biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281311(CHEMBL4159604)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575637(CHEMBL4845706)copy SMILES
Affinity DataIC50: 2nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281304(CHEMBL4160008)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone deacetylase 3(Homo sapiens (Human))TBA
LigandPNGBDBM29589(Faridak | LBH-589 | LBH-589B | Panobinostat | US10...)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of recombinant HDAC3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM29589(Faridak | LBH-589 | LBH-589B | Panobinostat | US10...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50442103(CHEMBL2441082)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281303(CHEMBL4171233)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281296(CHEMBL4173626)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575609(CHEMBL4852593)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575639(CHEMBL4858828)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575638(CHEMBL4847870)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575636(CHEMBL4848955)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 6(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Inhibition of full length human N-terminal GST-tagged HDAC6 using fluorogenic acetylated peptide as substrate incubated for 30 mins by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMedDrugBank
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575621(CHEMBL4865830)copy SMILES
Affinity DataIC50: 4nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
LigandPNGBDBM50105327(JNJ-26481585 | Quisinostat)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of C-terminal His-tagged recombinant human HDAC3 (1 to 428 residues)/N-terminal GST-tagged recombinant human NCoR2 (395 to 489 residues) c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
LigandPNGBDBM50575609(CHEMBL4852593)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of full length human C-terminal His-tagged HDAC3/human N-terminal GST-agged NCOR2 using fluorogenic acetylated peptide as substrate incuba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575640(CHEMBL4850570)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575623(CHEMBL4876993)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281298(CHEMBL4173668)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281281(CHEMBL4163369)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281307(CHEMBL4163329)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281321(CHEMBL4173662)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575621(CHEMBL4865830)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575642(CHEMBL4854765)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575624(CHEMBL4856110)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575636(CHEMBL4848955)copy SMILES
Affinity DataIC50: 7.20nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281297(CHEMBL4170114)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50281297(CHEMBL4170114)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X895VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50457746(CHEMBL4208004)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of G9a (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50575610(CHEMBL4872188)copy SMILES
Affinity DataIC50: 9nMAssay Description:Inhibition of full length human C-terminal His-tagged/C-terminal Flag-tagged HDAC1 using fluorogenic acetylated peptide as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575624(CHEMBL4856110)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575625(CHEMBL4862662)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575626(CHEMBL4876823)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575627(CHEMBL4863394)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575628(CHEMBL4862781)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575629(CHEMBL4855823)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575630(CHEMBL4870578)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575631(CHEMBL4869419)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575632(CHEMBL4874514)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575633(CHEMBL4855461)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575634(CHEMBL4856550)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575635(CHEMBL4854659)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575637(CHEMBL4845706)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias

Curated by ChEMBL
LigandPNGBDBM50575638(CHEMBL4847870)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human G9a enzyme using histone monomethyl-H3K9 peptide as substrate incubated for 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9V8VPubMed
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