Compile Data Set for Download or QSAR
Found 54 with Last Name = 'yanagisawa' and Initial = 'a'
LigandPNGBDBM50590513(CHEMBL5170356)copy SMILES
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590497(CHEMBL5182987)copy SMILES
Affinity DataIC50: 15nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590511(CHEMBL5175794)copy SMILES
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50603228(CHEMBL5194399)copy SMILES
Affinity DataIC50: 33nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603226(CHEMBL5189512)copy SMILES
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50590509(CHEMBL5188991)copy SMILES
Affinity DataIC50: 43nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590512(CHEMBL5173115)copy SMILES
Affinity DataIC50: 61nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590498(CHEMBL5171732)copy SMILES
Affinity DataIC50: 64nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50590498(CHEMBL5171732)copy SMILES
Affinity DataIC50: 64nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590507(CHEMBL5206581)copy SMILES
Affinity DataIC50: 71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50603229(CHEMBL5172873)copy SMILES
Affinity DataIC50: 83nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603218(CHEMBL5209124)copy SMILES
Affinity DataIC50: 87nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603225(CHEMBL5174328)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50590503(CHEMBL5202364)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590502(CHEMBL5206927)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590505(CHEMBL5193730)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590506(CHEMBL5187558)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590504(CHEMBL5196753)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50603224(CHEMBL5192802)copy SMILES
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50590510(CHEMBL5172080)copy SMILES
Affinity DataIC50: 103nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590496(CHEMBL5174202)copy SMILES
Affinity DataIC50: 120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590496(CHEMBL5174202)copy SMILES
Affinity DataIC50: 120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603221(CHEMBL5203083)copy SMILES
Affinity DataIC50: 249nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50590508(CHEMBL5188788)copy SMILES
Affinity DataIC50: 288nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50603227(CHEMBL5208550)copy SMILES
Affinity DataIC50: 315nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603222(CHEMBL5194891)copy SMILES
Affinity DataIC50: 354nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603220(CHEMBL5205017)copy SMILES
Affinity DataIC50: 404nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603219(CHEMBL5198191)copy SMILES
Affinity DataIC50: 455nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50590496(CHEMBL5174202)copy SMILES
Affinity DataIC50: 838nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50603223(CHEMBL5188634)copy SMILES
Affinity DataIC50: 997nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7TXQPubMed
LigandPNGBDBM50590501(CHEMBL5180294)copy SMILES
Affinity DataIC50: 1.14E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590500(CHEMBL5180542)copy SMILES
Affinity DataIC50: 1.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
LigandPNGBDBM50590499(CHEMBL5169559)copy SMILES
Affinity DataIC50: 2.88E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2N4KPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469403(CHEMBL4285849)copy SMILEScopy InChI
Affinity DataEC50:  593nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469402(CHEMBL4288363)copy SMILEScopy InChI
Affinity DataEC50:  13nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469401(CHEMBL4289449)copy SMILEScopy InChI
Affinity DataEC50:  84nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50093473(Arhalofenate | CB-102 | JNJ-39659100 | M-102 | MBX...)copy SMILEScopy InChI
Affinity DataEC50: >500nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as cell differentiation after 5 days by Hoechst 33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469400(CHEMBL4278109)copy SMILEScopy InChI
Affinity DataEC50:  2.40nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469398(ATx08-001 | FK-614)copy SMILEScopy InChI
Affinity DataEC50:  163nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469399(CHEMBL4293061)copy SMILEScopy InChI
Affinity DataEC50:  57nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469398(ATx08-001 | FK-614)copy SMILEScopy InChI
Affinity DataEC50: >500nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as cell differentiation after 5 days by Hoechst 33342 staining-based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50093473(Arhalofenate | CB-102 | JNJ-39659100 | M-102 | MBX...)copy SMILEScopy InChI
Affinity DataEC50:  7.37E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50103521(Actos | CHEBI:8228 | Duetact | Pioglitazone | US10...)copy SMILEScopy InChI
Affinity DataEC50:  2.05E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469397(CHEMBL4277928)copy SMILEScopy InChI
Affinity DataEC50:  151nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469396(CHEMBL4282451)copy SMILEScopy InChI
Affinity DataEC50:  166nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469395(CHEMBL4277723)copy SMILEScopy InChI
Affinity DataEC50:  33nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469394(CHEMBL4286027)copy SMILEScopy InChI
Affinity DataEC50:  2.70nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469393(CHEMBL4281564)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50469392(CHEMBL4289861)copy SMILEScopy InChI
Affinity DataEC50:  177nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DXVPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Fuji Research Park, R&D Division

Curated by ChEMBL
LigandPNGBDBM50428854(CHEMBL1236924)copy SMILEScopy InChI
Affinity DataEC50:  59nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Displayed 1 to 50 (of 54 total ) | Next | Last >>
Jump to: