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Found 467 with Last Name = 'samatar' and Initial = 'aa'
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103302(SCH772984 | US8546404, 6)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2959G61US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50094464(CHEMBL3590107 | US10525036, Example SCH772984 | US...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of ERK2 (unknown origin) preincubated for 45 mins followed by substrate addition measured after 0.5 hrs by IMAP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50094464(CHEMBL3590107 | US10525036, Example SCH772984 | US...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50458811(CHEMBL4209570)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1G9SPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579208(CHEMBL4867107)copy SMILES
Affinity DataIC50: 2nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103295(US8546404, 462)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2959G61US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM103295(US8546404, 462)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JW8PubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579222(CHEMBL4861383)copy SMILES
Affinity DataIC50: 2.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518531(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518527(2-Alyl-6-((2′,3′-dihydro-1′H-spi...)copy SMILES
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518526(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518538(2-Allyl-6-((2-(2-hydroxyethyl)-1,2,3,4-tetrahydroi...)copy SMILES
Affinity DataIC50: 2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103292(US8546404, 1729 | US8546404, 469)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2959G61US Patent
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM34531(US8546404, 459)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2959G61US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579228(CHEMBL4867211)copy SMILES
Affinity DataIC50: 2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103292(US8546404, 1729 | US8546404, 469)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2959G61US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518540(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579214(CHEMBL4856035)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579225(CHEMBL4874546)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518530(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579218(CHEMBL4876612)copy SMILES
Affinity DataIC50: 2.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579223(CHEMBL4853285)copy SMILES
Affinity DataIC50: 3.10nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579224(CHEMBL4861351)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579227(CHEMBL4847705)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579221(CHEMBL4866800)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579216(CHEMBL4865963)copy SMILES
Affinity DataIC50: 3.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579213(CHEMBL4853973)copy SMILES
Affinity DataIC50: 3.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579220(CHEMBL4868683)copy SMILES
Affinity DataIC50: 3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579219(CHEMBL4857841)copy SMILES
Affinity DataIC50: 3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579215(CHEMBL4861168)copy SMILES
Affinity DataIC50: 4.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103293(US8546404, 480)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2959G61US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579211(CHEMBL4871803)copy SMILES
Affinity DataIC50: 4.80nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM103293(US8546404, 480)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JW8PubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50458805(CHEMBL4206960)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1G9SPubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50458806(CHEMBL4205192)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1G9SPubMed
TargetMitogen-activated protein kinase 1(Mus musculus (Mouse))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM103296(US8546404, 622)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Activated ERK2 activity was determined in the IMAP assay format.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2959G61US Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579212(CHEMBL4879157)copy SMILES
Affinity DataIC50: 5.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50461920(CHEMBL4225841)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JW8PubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50458802(CHEMBL4215228)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50458802(CHEMBL4215228)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579210(CHEMBL4853185)copy SMILES
Affinity DataIC50: 5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579210(CHEMBL4853185)copy SMILES
Affinity DataIC50: 5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50461917(CHEMBL4225054)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JW8PubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50458807(CHEMBL4216900)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1G9SPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579209(CHEMBL4874090)copy SMILES
Affinity DataIC50: 6.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM103297(US8546404, 613)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1G9SPubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM103297(US8546404, 613)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of ERK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JW8PubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Merck & Co.

Curated by ChEMBL
LigandPNGBDBM50458803(CHEMBL4213970)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of ERK2 (unknown origin) using peptide substrate measured after 45 mins by IMAP assayMore data for this Ligand-Target Pair
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