Compile Data Set for Download or QSAR
Found 59 with Last Name = 'goldberg' and Initial = 'afg'
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562854(CHEMBL4763993)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562860(CHEMBL4762311)copy SMILES
Affinity DataIC50: 600nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562857(CHEMBL4791813)copy SMILES
Affinity DataIC50: 700nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562869(CHEMBL4759891)copy SMILES
Affinity DataIC50: 900nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562861(CHEMBL4792077)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50561073(CHEMBL4751295)copy SMILES
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562864(CHEMBL4756916)copy SMILES
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562860(CHEMBL4762311)copy SMILES
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50155928(3,4-Methylenedioxyb-Nitrostyrene | CHEMBL596380)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50155928(3,4-Methylenedioxyb-Nitrostyrene | CHEMBL596380)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50561073(CHEMBL4751295)copy SMILES
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562859(CHEMBL4742209)copy SMILES
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562859(CHEMBL4742209)copy SMILES
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50532921(CHEMBL594404)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562863(CHEMBL4788535)copy SMILES
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50249208(2-methoxy-4-(2-nitrovinyl)phenyl benzoate | CHEMBL...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562868(CHEMBL4790925)copy SMILES
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562858(CHEMBL2409306)copy SMILES
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562864(CHEMBL4756916)copy SMILES
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562858(CHEMBL2409306)copy SMILES
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562868(CHEMBL4790925)copy SMILES
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562857(CHEMBL4791813)copy SMILES
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562863(CHEMBL4788535)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50532921(CHEMBL594404)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562856(CHEMBL4763795)copy SMILES
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562854(CHEMBL4763993)copy SMILES
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562855(CHEMBL4763517)copy SMILES
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562865(CHEMBL4795080)copy SMILES
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50514012(CHEMBL3220938)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50248767(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562856(CHEMBL4763795)copy SMILES
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562862(CHEMBL4752271)copy SMILES
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562861(CHEMBL4792077)copy SMILES
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562855(CHEMBL4763517)copy SMILES
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50249208(2-methoxy-4-(2-nitrovinyl)phenyl benzoate | CHEMBL...)copy SMILEScopy InChI
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50248767(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562869(CHEMBL4759891)copy SMILES
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50007082((E)-2-methoxy-4-(2-nitrovinyl)phenol | 2-Methoxy-4...)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562865(CHEMBL4795080)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50324690(CHEMBL1221767 | N-(4-((1,1'-biphenyl)-4-ylamino)qu...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50007082((E)-2-methoxy-4-(2-nitrovinyl)phenol | 2-Methoxy-4...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50324690(CHEMBL1221767 | N-(4-((1,1'-biphenyl)-4-ylamino)qu...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM123747(1-(tert-butyl)-3-phenyl-1H-pyrazolo[3,4-d]pyrimidi...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50486070(3,4-(Methylenedioxy)Cinnamic Acid | 3,4-Methylened...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50248765(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50486070(3,4-(Methylenedioxy)Cinnamic Acid | 3,4-Methylened...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562867(CHEMBL4757121)copy SMILES
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50514012(CHEMBL3220938)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of His6-tagged p97 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in ATPase activity measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50562866(CHEMBL4749210)copy SMILES
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
TargetTransitional endoplasmic reticulum ATPase(Homo sapiens (Human))TBA
LigandPNGBDBM50345704(1-(tert-butyl)-3-(naphthalen-2-yl)-1H-pyrazolo[3,4...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of p97 in human HeLa cells assessed as reduction in proteasomal turnover of p97-dependent reporter substrate UbG76V-GFP incubated for 120 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2T24PubMed
Displayed 1 to 50 (of 59 total ) | Next | Last >>
Jump to: