Compile Data Set for Download or QSAR
Found 207 with Last Name = 'wright' and Initial = 'ag'
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437403(CHEMBL2408771)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427749(CHEMBL2324924)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437403(CHEMBL2408771)copy SMILEScopy InChI
Affinity DataIC50: 0.270nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427748(CHEMBL2324925)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427749(CHEMBL2324924)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50228407(8-((R)-3-amino-piperidin-1-yl)-3-methyl-7-(3-methy...)copy SMILEScopy InChI
Affinity DataIC50: 0.730nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427749(CHEMBL2324924)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50228407(8-((R)-3-amino-piperidin-1-yl)-3-methyl-7-(3-methy...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437404(CHEMBL2408655)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427748(CHEMBL2324925)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427747(CHEMBL2324926)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427749(CHEMBL2324924)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50228407(8-((R)-3-amino-piperidin-1-yl)-3-methyl-7-(3-methy...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437403(CHEMBL2408771)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437404(CHEMBL2408655)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427750(CHEMBL2324923)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of wild type Abl1 kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427749(CHEMBL2324924)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427750(CHEMBL2324923)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427748(CHEMBL2324925)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetSerine protease hepsin(Homo sapiens (Human))
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant C-terminal His10-tagged human Hepsin (R45 to L17 residues) D161E/ R162K double mutant expressed in mouse NS0 cells using Bo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3VVTPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427747(CHEMBL2324926)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437395(CHEMBL2408638)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427748(CHEMBL2324925)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427742(CHEMBL2324930)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437404(CHEMBL2408655)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437395(CHEMBL2408638)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427748(CHEMBL2324925)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427750(CHEMBL2324923)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437404(CHEMBL2408655)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of human DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427745(CHEMBL2324927)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427747(CHEMBL2324926)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427750(CHEMBL2324923)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427741(CHEMBL2324931)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427744(CHEMBL2324928)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427750(CHEMBL2324923)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427742(CHEMBL2324930)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437396(CHEMBL2408651)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437396(CHEMBL2408651)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetDipeptidyl peptidase 4(Sus scrofa (pig))
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437402(CHEMBL2408774)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HQ41BXPubMed
TargetTyrosine-protein kinase ABL2(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427741(CHEMBL2324931)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of Abl2 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427743(CHEMBL2324929)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetSerine protease hepsin(Homo sapiens (Human))
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50272185(CHEMBL4129836)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant C-terminal His10-tagged human Hepsin (R45 to L17 residues) D161E/ R162K double mutant expressed in mouse NS0 cells using Bo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3VVTPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427747(CHEMBL2324926)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of P38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medicine

Curated by ChEMBL
LigandPNGBDBM50530609(CHEMBL4461010)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human 20S proteasome subunit beta-5i using Ac-ANW-AMC as substrate and measured every 30 secs for 30 mins by microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M695MPubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Weill Cornell Medicine

Curated by ChEMBL
LigandPNGBDBM50530609(CHEMBL4461010)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human 20S proteasome subunit beta-5i using Ac-ANW-AMC as substrate and measured every 30 secs for 30 mins by microtiter plate assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M695MPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427747(CHEMBL2324926)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427741(CHEMBL2324931)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetSerine protease hepsin(Homo sapiens (Human))
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50424712(CAMOSTAT | Camostat Mesilate | Foipan)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant C-terminal His10-tagged human Hepsin (R45 to L17 residues) D161E/ R162K double mutant expressed in mouse NS0 cells using Bo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3VVTPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427745(CHEMBL2324927)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Cyclofluidic Ltd

Curated by ChEMBL
LigandPNGBDBM50427744(CHEMBL2324928)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of Abl1 kinase (unknown origin) using Tyr 6 peptide as substrate assessed as residual enzyme activity after every 10 secs measured for 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6KPDPubMed
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