Found 89 with Last Name = 'hassan' and Initial = 'ahe' TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataKi: 129nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
TargetDeath-associated protein kinase 1(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataKi: 581nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of red tracer binding to human ERG expressed in membranes preincubated for 10 to 15 mins followed by tracer addition measured after 3 hrs ...More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of 1 uM [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 204nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 219nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 219nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 245nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 252nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured after 60 minsMore data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 273nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of 100 uM [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
Affinity DataIC50: 288nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 299nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured after 40 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 347nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 347nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 372nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured immediatelyMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 575nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate incubated for 10 mins followed by substrate addition and me...More data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
TargetDeath-associated protein kinase 1(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 100 uM [gamma-33P]-ATP by filtration met...More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Displacement of [3H]CP55940 from membrane bound human CB2 receptor after 1 hr by beta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Irreversible inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate measured immediatelyMore data for this Ligand-Target Pair
TargetDeath-associated protein kinase 1(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of human DAPK1 (1 to 363 residues) using KKLNRTLSFAEPG as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration meth...More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Displacement of [3H]SR141716A from membrane bound human CB1 receptor after 1 hr by beta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+3nMAssay Description:Displacement of [3H]CP55940 from membrane bound human CB2 receptor after 1 hr by beta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of IKKbeta (unknown origin) using IkappaBalpha-derived 5FAMGRHDSGLDSMK-NH2 as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 1.71E+3nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Korea Institute of Science and Technology (KIST)
Curated by ChEMBL
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of human CSF1R using poly[Glu:Tyr] (4:1) as substrate after 120 mins in presence of 10 uM [gamma-33P]-ATP by filtration methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.43E+3nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 2.61E+3nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
Affinity DataIC50: 2.61E+3nMAssay Description:Allosteric inhibition of IKKbeta (unknown origin) using 5FAM-GRHDSGLDSMK-NH2 as substrate pretreated for 10 mins followed measured after 2 hrs by TR-...More data for this Ligand-Target Pair
