Compile Data Set for Download or QSAR
Found 228 with Last Name = 'kwong' and Initial = 'aj'
LigandPNGBDBM50434072(CHEMBL2381342)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of MEK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM50559800(CHEMBL3329977)copy SMILES
Affinity DataIC50: 1.90nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM50559802(CHEMBL4303171)copy SMILES
Affinity DataIC50: 4.30nMAssay Description:Inhibition of MEK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM50553870(CHEMBL4749823)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM50206444(CHEMBL3901151)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM50615119(CHEMBL5284723)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50559801(CHEMBL4787266)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)copy SMILES
Affinity DataIC50: 41nMAssay Description:Inhibition of MEK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)copy SMILES
Affinity DataIC50: 41nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50615123(CHEMBL5283781)copy SMILES
Affinity DataIC50: 42nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50615102(CHEMBL5271442)copy SMILES
Affinity DataIC50: 60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM558862(US11370770, Compound 6n)copy SMILES
Affinity DataIC50: 60nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50577661(CHEMBL4879048)copy SMILES
Affinity DataIC50: 61nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50MCPubMed
LigandPNGBDBM558880(US11370770, Compound 6ee)copy SMILES
Affinity DataIC50: 63nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50615113(CHEMBL5267499)copy SMILES
Affinity DataIC50: 66nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)copy SMILES
Affinity DataIC50: 66nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50615120(CHEMBL5279577)copy SMILES
Affinity DataIC50: 74nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50577689(CHEMBL4866649)copy SMILES
Affinity DataIC50: 83nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50MCPubMed
LigandPNGBDBM50577657(CHEMBL4848865)copy SMILES
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50MCPubMed
LigandPNGBDBM50577689(CHEMBL4866649)copy SMILES
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK7 expressed in Sf21 cells using JNK1 as substrate pre-incubated for 30 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50MCPubMed
LigandPNGBDBM558875(US11370770, Compound 6z)copy SMILES
Affinity DataIC50: 100nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50559798(CHEMBL4758063 | US11370770, Compound 6ff)copy SMILES
Affinity DataIC50: 100nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558864(US11370770, Compound 6p)copy SMILES
Affinity DataIC50: 110nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50615118(CHEMBL5271266)copy SMILES
Affinity DataIC50: 110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50615122(CHEMBL5267684)copy SMILES
Affinity DataIC50: 110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM558878(US11370770, Compound 6cc)copy SMILES
Affinity DataIC50: 120nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558862(US11370770, Compound 6n)copy SMILES
Affinity DataIC50: 130nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558867(US11370770, Compound 6s)copy SMILES
Affinity DataIC50: 150nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558848(US11370770, Compound 6a)copy SMILES
Affinity DataIC50: 180nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558867(US11370770, Compound 6s)copy SMILES
Affinity DataIC50: 180nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50559799(CHEMBL4748767)copy SMILES
Affinity DataIC50: 190nMAssay Description:Inhibition of MEK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM558866(US11370770, Compound 6r)copy SMILES
Affinity DataIC50: 200nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558865(US11370770, Compound 6q)copy SMILES
Affinity DataIC50: 210nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558867(US11370770, Compound 6s)copy SMILES
Affinity DataIC50: 220nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50504351(CHEMBL100206)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of MEK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028W77PubMed
LigandPNGBDBM558858(US11370770, Compound 6j)copy SMILES
Affinity DataIC50: 240nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558858(US11370770, Compound 6j)copy SMILES
Affinity DataIC50: 250nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50615109(CHEMBL5282673)copy SMILES
Affinity DataIC50: 260nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM558880(US11370770, Compound 6ee)copy SMILES
Affinity DataIC50: 260nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50615129(CHEMBL5277855)copy SMILES
Affinity DataIC50: 260nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM31085(1-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 260nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50615110(CHEMBL5271906)copy SMILES
Affinity DataIC50: 270nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50577686(CHEMBL4865159)copy SMILES
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50MCPubMed
LigandPNGBDBM50615128(CHEMBL5272546)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50577671(CHEMBL4872723)copy SMILES
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50MCPubMed
LigandPNGBDBM50577647(CHEMBL4849172)copy SMILES
Affinity DataIC50: 310nMAssay Description:Inhibition of human recombinant full length N-terminal GST tagged MEK4 expressed in Sf21 cells using p38 alpha as substrate pre-incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50MCPubMed
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))TBA
LigandPNGBDBM558875(US11370770, Compound 6z)copy SMILES
Affinity DataIC50: 350nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM50615121(CHEMBL5271334)copy SMILES
Affinity DataIC50: 360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50615130(CHEMBL5271519)copy SMILES
Affinity DataIC50: 360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM558875(US11370770, Compound 6z)copy SMILES
Affinity DataIC50: 360nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
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