Compile Data Set for Download or QSAR
Found 196 with Last Name = 'cecil' and Initial = 'ar'
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM19152((1S,7R,10S,16E,21R)-21-methyl-7-(propan-2-yl)-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMpH: 8.0 T: 2°CAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N4BPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM19153((1S,7R,10S,16E,21R)-7,21-bis(propan-2-yl)-2-oxa-12...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMpH: 8.0 T: 2°CAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N4BPubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM310701(US10150763, Example A)copy SMILEScopy InChI
Affinity DataIC50: 1.76nMAssay Description:The assay is described in WO2008/062201.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C82CC1US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM19151((1S,4S,7Z,10S,16E,21R)-7-ethylidene-4,21-bis(propa...)copy SMILEScopy InChI
Affinity DataIC50: 3.97nMpH: 8.0 T: 2°CAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N4BPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM136702(US8865655, 10)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMT: 2°CAssay Description:In vitro HDAC assays were performed using a HDAC fluorescent activity assay kit (Biomol, UK) according to the manufacturer's instructions. Compounds ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Z036V4US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291359((E)-3-[2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291359((E)-3-[2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291360(US9580442, Example H | US9938290, H | [2-(1H-Indol...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291363(2-(1H-Indol-4-yl)-4-morpholin-4-yl-8-morpholin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291355(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291355(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291358((E)-1-(4-Methyl-piperazin-1-yl)-3-[4-morpholin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291360(US9580442, Example H | US9938290, H | [2-(1H-Indol...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291363(2-(1H-Indol-4-yl)-4-morpholin-4-yl-8-morpholin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM387173(US9938290, F)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291357(2,8-Bis-(1H-indol-4-yl)-4-morpholin-4-yl-pyrido[3&...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291357(2,8-Bis-(1H-indol-4-yl)-4-morpholin-4-yl-pyrido[3&...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291365(2-(1H-Indol-4-yl)-4,8-di-morpholin-4-yl-pyrido[3&#...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291361(2-(1H-Indol-4-yl)-4-morpholin-4-yl-8-piperidin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291365(2-(1H-Indol-4-yl)-4,8-di-morpholin-4-yl-pyrido[3&#...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291361(2-(1H-Indol-4-yl)-4-morpholin-4-yl-8-piperidin-1-y...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291354(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291354(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM19154((6R,9R,12R,16R)-9,12-dimethyl-6-(propan-2-yl)-16-[...)copy SMILEScopy InChI
Affinity DataIC50: 17.5nMpH: 8.0 T: 2°CAssay Description:For the enzyme assay, the enzyme fraction was added to fluorescent substrate in the presence of test compounds, and the mixture was incubated for add...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7N4BPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291355(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291355(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291364(US9580442, Example L | US9938290, L | [2-(1H-Indol...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291364(US9580442, Example L | US9938290, L | [2-(1H-Indol...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM136703(US8865655, 11)copy SMILEScopy InChI
Affinity DataIC50: 21.6nMT: 2°CAssay Description:In vitro HDAC assays were performed using a HDAC fluorescent activity assay kit (Biomol, UK) according to the manufacturer's instructions. Compounds ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Z036V4US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291366(3-{4-[2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3&...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291366(3-{4-[2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3&...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291365(2-(1H-Indol-4-yl)-4,8-di-morpholin-4-yl-pyrido[3&#...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291365(2-(1H-Indol-4-yl)-4,8-di-morpholin-4-yl-pyrido[3&#...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291362(2-(1H-Indol-4-yl)-8-(4-methyl-piperazin-1-ylmethyl...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291362(2-(1H-Indol-4-yl)-8-(4-methyl-piperazin-1-ylmethyl...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291356(4-Morpholin-4-yl-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291356(4-Morpholin-4-yl-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Southampton

LigandPNGBDBM136704(US8865655, 16)copy SMILEScopy InChI
Affinity DataIC50: 47nMT: 2°CAssay Description:In vitro HDAC assays were performed using a HDAC fluorescent activity assay kit (Biomol, UK) according to the manufacturer's instructions. Compounds ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Z036V4US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291354(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Lek Pharmaceuticals d.d.

LigandPNGBDBM291354(2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3′...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291356(4-Morpholin-4-yl-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291356(4-Morpholin-4-yl-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291360(US9580442, Example H | US9938290, H | [2-(1H-Indol...)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291360(US9580442, Example H | US9938290, H | [2-(1H-Indol...)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291363(2-(1H-Indol-4-yl)-4-morpholin-4-yl-8-morpholin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291363(2-(1H-Indol-4-yl)-4-morpholin-4-yl-8-morpholin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291357(2,8-Bis-(1H-indol-4-yl)-4-morpholin-4-yl-pyrido[3&...)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291357(2,8-Bis-(1H-indol-4-yl)-4-morpholin-4-yl-pyrido[3&...)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291359((E)-3-[2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3...)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:PI3K Isoform using biochemical assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VM2US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Karus Therapeutics Limited

US Patent
LigandPNGBDBM291359((E)-3-[2-(1H-Indol-4-yl)-4-morpholin-4-yl-pyrido[3...)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Please see articleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5H9PUS Patent
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