Compile Data Set for Download or QSAR
Found 20 with Last Name = 'sørensen' and Initial = 'ar'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130727(1-(4-Amino-furazan-3-yl)-5-pyrrolidin-1-ylmethyl-1...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130724(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130732(4-[4-(5-Pyridin-4-yl-4H-[1,2,4]triazol-3-yl)-5-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130719(4-[5-Piperidin-1-ylmethyl-4-(5-pyridin-4-yl-4H-[1,...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130725(3-(3-Chloro-4-hydroxy-phenylamino)-4-(2-nitro-phen...)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130725(3-(3-Chloro-4-hydroxy-phenylamino)-4-(2-nitro-phen...)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130730(1-(4-Amino-furazan-3-yl)-5-diethylaminomethyl-1H-[...)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130720(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130726(1-(4-Amino-furazan-3-yl)-5-pyrrolidin-1-ylmethyl-1...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130722(4-[5-Dimethylaminomethyl-4-(5-pyridin-4-yl-4H-[1,2...)copy SMILEScopy InChI
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130733(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130731(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130728(1-(4-Amino-furazan-3-yl)-5-diethylaminomethyl-1H-[...)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130721(1-(4-Amino-furazan-3-yl)-5-diethylaminomethyl-1H-[...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human Glycogen synthase kinase-3 beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130724(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130720(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130719(4-[5-Piperidin-1-ylmethyl-4-(5-pyridin-4-yl-4H-[1,...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of Cyclin-dependent kinase 2-cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130723(1-(4-Amino-furazan-3-yl)-5-piperidin-1-ylmethyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50130729(1-(4-Amino-furazan-3-yl)-5-(isobutylamino-methyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibitory activity against human glycogen synthase kinase-3beta (GSK3-beta) at 100 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76D9BPubMed