Compile Data Set for Download or QSAR
Found 327 with Last Name = 'hung' and Initial = 'aw'
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455611(CHEMBL4212424)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455569(CHEMBL4202753)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455593(CHEMBL4208685)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455592(CHEMBL4206065)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455602(CHEMBL4216507)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455589(CHEMBL4213984)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-zeta expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520279(CHEMBL4442209)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520278(CHEMBL4569209)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM31085(1-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of MNK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455566(CHEMBL4208028)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520279(CHEMBL4442209)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520296(CHEMBL4588193)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520256(CHEMBL4443472)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455611(CHEMBL4212424)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455611(CHEMBL4212424)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455589(CHEMBL4213984)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520278(CHEMBL4569209)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520292(CHEMBL4462099)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520252(CHEMBL4440223)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455593(CHEMBL4208685)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455594(CHEMBL4212934)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455569(CHEMBL4202753)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520289(CHEMBL4587472)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520296(CHEMBL4588193)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520253(CHEMBL4587832)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50172078(LY-2801653 | Merestinib)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Inhibition of MNK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455602(CHEMBL4216507)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455610(CHEMBL4211722)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520252(CHEMBL4440223)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520256(CHEMBL4443472)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455588(CHEMBL4208982)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520292(CHEMBL4462099)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50172078(LY-2801653 | Merestinib)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of MNK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455592(CHEMBL4206065)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520276(CHEMBL4457274)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1/2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520279(CHEMBL4442209)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of MNK1/MNK2 in human HeLa cells overexpressing eIF4E assessed as reduction in eIF4E phosphorylation at Ser209 residue after 2 hrs by Alph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455593(CHEMBL4208685)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1/2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520253(CHEMBL4587832)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of MNK1/MNK2 in human HeLa cells overexpressing eIF4E assessed as reduction in eIF4E phosphorylation at Ser209 residue after 2 hrs by Alph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520253(CHEMBL4587832)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455602(CHEMBL4216507)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455566(CHEMBL4208028)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50526595(CHEMBL4517782)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant human full length N-terminal GST-fused PKCi (1 to 587 residues) expressed in baculovirus expression system using 5-FAM-RFAR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348PT0PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455589(CHEMBL4213984)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455568(CHEMBL4215492)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V69N5ZPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))TBA
LigandPNGBDBM50578087(CHEMBL4871523)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of Axl (unknown origin) using 5'FAM labeled KKKKEEIYFFF-NH2 peptide as substrate incubated for 1.5 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70KN7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520270(CHEMBL4456135)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520261(CHEMBL4558635)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of N-terminal GST-tagged MNK2 (unknown origin) (72 to 385 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520289(CHEMBL4587472)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of N-terminal GST-tagged MNK1 (unknown origin) (37 to 341 residues) expressed in Escherichia coli BL21 (DE3) cells using 5-FAM-TATKSGSTTKN...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1/2(Homo sapiens (Human))
A*STAR

Curated by ChEMBL
LigandPNGBDBM50520278(CHEMBL4569209)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of MNK1/MNK2 in human HeLa cells overexpressing eIF4E assessed as reduction in eIF4E phosphorylation at Ser209 residue after 2 hrs by Alph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27084T7PubMed
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50526582(CHEMBL4471416)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant human full length N-terminal GST-fused PKCi (1 to 587 residues) expressed in baculovirus expression system using 5-FAM-RFAR...More data for this Ligand-Target Pair
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