Compile Data Set for Download or QSAR
Found 78 with Last Name = 'chan' and Initial = 'awe'
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541233(CHEMBL4638227)copy SMILEScopy InChI
Affinity DataIC50: 101nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541238(CHEMBL4641181)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541237(CHEMBL4641186)copy SMILEScopy InChI
Affinity DataIC50: 176nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50350236(CHEMBL1812335)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541234(CHEMBL4642040)copy SMILEScopy InChI
Affinity DataIC50: 232nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541236(CHEMBL4635348)copy SMILEScopy InChI
Affinity DataIC50: 258nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541235(CHEMBL4640878)copy SMILEScopy InChI
Affinity DataIC50: 259nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetNeuropilin-1(Homo sapiens (Human))
NCE Discovery (Domainex Ltd

Curated by ChEMBL
LigandPNGBDBM50453006(CHEMBL4217624)copy SMILEScopy InChI
Affinity DataIC50: 609nMAssay Description:Inhibition of biotinylated VEGF-A binding to N-terminal His6-tagged recombinant human NRP1-b1 domain expressed in Escherichia coli Rosetta Gami 2 (DE...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81GNKPubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541228(CHEMBL4634649)copy SMILEScopy InChI
Affinity DataIC50: 970nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541212(CHEMBL4633506)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541225(CHEMBL4633533)copy SMILEScopy InChI
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetNeuropilin-1(Homo sapiens (Human))
NCE Discovery (Domainex Ltd

Curated by ChEMBL
LigandPNGBDBM50453006(CHEMBL4217624)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of biotinylated VEGF-A binding to human NRP1 expressed in human DU145 cells after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q81GNKPubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541229(CHEMBL4639748)copy SMILEScopy InChI
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541230(CHEMBL4645791)copy SMILEScopy InChI
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541209(CHEMBL4649787)copy SMILEScopy InChI
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541226(CHEMBL4645162)copy SMILEScopy InChI
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541224(CHEMBL4634256)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541218(CHEMBL4638376)copy SMILEScopy InChI
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541223(CHEMBL4648086)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541227(CHEMBL4635718)copy SMILEScopy InChI
Affinity DataIC50: 3.85E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541214(CHEMBL4645826)copy SMILEScopy InChI
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541219(CHEMBL4642580)copy SMILEScopy InChI
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554127(CHEMBL4756598)copy SMILES
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541232(CHEMBL4634340)copy SMILEScopy InChI
Affinity DataIC50: 8.76E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541233(CHEMBL4638227)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541231(CHEMBL4641346)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541213(CHEMBL4642931)copy SMILEScopy InChI
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541210(CHEMBL4637427)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541217(CHEMBL4634329)copy SMILEScopy InChI
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541222(CHEMBL4644336)copy SMILEScopy InChI
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554128(CHEMBL4750759)copy SMILES
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541215(CHEMBL4641495)copy SMILEScopy InChI
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541220(CHEMBL4647738)copy SMILEScopy InChI
Affinity DataIC50: 2.53E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541233(CHEMBL4638227)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541233(CHEMBL4638227)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541221(CHEMBL4633689)copy SMILEScopy InChI
Affinity DataIC50: 7.64E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554126(CHEMBL4777408)copy SMILES
Affinity DataIC50: 8.30E+4nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554126(CHEMBL4777408)copy SMILES
Affinity DataIC50: 1.17E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in absence of DTT by [gamma-33P]-AT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554129(CHEMBL4752126)copy SMILES
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541216(CHEMBL4633276)copy SMILEScopy InChI
Affinity DataIC50: 4.10E+5nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554118(CHEMBL4794430)copy SMILES
Affinity DataIC50: 4.20E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554123(CHEMBL4783213)copy SMILES
Affinity DataIC50: 4.30E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554121(CHEMBL4745854)copy SMILES
Affinity DataIC50: 4.97E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554122(CHEMBL4742648)copy SMILES
Affinity DataIC50: 5.42E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50541211(CHEMBL4647039)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+5nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S35PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554126(CHEMBL4777408)copy SMILES
Affinity DataIC50: 7.31E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence of DTT by [gamma-33P]-A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554120(CHEMBL4754114)copy SMILES
Affinity DataIC50: 9.10E+5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554119(CHEMBL4792773)copy SMILES
Affinity DataIC50: 1.10E+6nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554117(CHEMBL4756152)copy SMILES
Affinity DataIC50: 1.30E+6nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50554124(CHEMBL4748202)copy SMILES
Affinity DataIC50: 1.30E+6nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using myelin basic protein as substrate incubated for 30 mins in presence or absence of DTT by [g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0ZJ6PubMed
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