Compile Data Set for Download or QSAR
Found 143 with Last Name = 'bhushan' and Initial = 'b'
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273478(CHEMBL4130224)copy SMILEScopy InChI
Affinity DataKi:  7.40E+4nMAssay Description:Mixed type inhibition of KDM5A (L88 to G353 residues) ARID/PHD1/2/3 deletion mutant (unknown origin) demethylation activity using H3(1-21)K4me3 pepti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454844(CHEMBL4204694)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454844(CHEMBL4204694)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454854(CHEMBL4209038)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454854(CHEMBL4209038)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454848(CHEMBL4205285)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454855(CHEMBL4215000)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454853(CHEMBL4205183)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454859(CHEMBL4206181)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454849(CHEMBL4218675)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454849(CHEMBL4218675)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454855(CHEMBL4215000)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454859(CHEMBL4206181)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454858(CHEMBL4218774)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454848(CHEMBL4205285)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454846(CHEMBL4211201)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454847(CHEMBL4203936)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454853(CHEMBL4205183)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454847(CHEMBL4203936)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454858(CHEMBL4218774)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454846(CHEMBL4211201)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454856(CHEMBL4208277)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454845(CHEMBL4213743)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454857(CHEMBL4218482)copy SMILEScopy InChI
Affinity DataIC50: 82nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454845(CHEMBL4213743)copy SMILEScopy InChI
Affinity DataIC50: 151nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454857(CHEMBL4218482)copy SMILEScopy InChI
Affinity DataIC50: 154nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454852(CHEMBL4208111)copy SMILEScopy InChI
Affinity DataIC50: 164nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454850(CHEMBL4206582)copy SMILEScopy InChI
Affinity DataIC50: 173nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454850(CHEMBL4206582)copy SMILEScopy InChI
Affinity DataIC50: 208nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454856(CHEMBL4208277)copy SMILEScopy InChI
Affinity DataIC50: 269nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454852(CHEMBL4208111)copy SMILEScopy InChI
Affinity DataIC50: 373nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454851(CHEMBL4209558)copy SMILEScopy InChI
Affinity DataIC50: 466nMAssay Description:Inhibition of KDM4C (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454851(CHEMBL4209558)copy SMILEScopy InChI
Affinity DataIC50: 615nMAssay Description:Inhibition of KDM4A (unknown origin) expressed in Escherichia coli using biotinylated peptide as substrate pretreated for 15 mins followed by substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD435TPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM223320(KDOAM-25)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of KDM5A (M1 to L801 residues) PHD2/3 deletion mutant (unknown origin) demethylation activity preincubated for 10 mins followed by peptide...More data for this Ligand-Target Pair
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273472(CHEMBL4126235)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7B (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM223320(KDOAM-25)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of KDM5A (M1 to L801 residues) PHD2/3 deletion mutant (unknown origin) demethylation activity preincubated for 10 mins followed by peptide...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273472(CHEMBL4126235)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase PHF2(Homo sapiens)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273472(CHEMBL4126235)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7C (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50270477(CHEMBL4127210)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from recombinant His6-tagged human KDM5A (PHD3) (1542 to 1660 residues) ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92787(WAG-003)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of H3K4me3 binding to Halo-tagged GST-fused KDM5A PHD3 domain (unknown origin) expressed in Escherichia coli by HaloTag-based peptide di...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273478(CHEMBL4130224)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from recombinant His6-tagged human KDM5A (PHD3) (1542 to 1660 residues) ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92788(WAG-005)copy SMILEScopy InChI
Affinity DataIC50: 4.10E+4nMAssay Description:Displacement of H3K4me3 binding to Halo-tagged GST-fused KDM5A PHD3 domain (unknown origin) expressed in Escherichia coli by HaloTag-based peptide di...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92788(WAG-005)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92788(WAG-005)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273477(CHEMBL4129830)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273474(CHEMBL4129980)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273478(CHEMBL4130224)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of KDM5A (M1 to L801 residues) PHD2/3 deletion mutant (unknown origin) demethylation activity preincubated for 10 mins followed by peptide...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92788(WAG-005)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibition of KDM5A (M1 to L801 residues) PHD2/3 deletion mutant (unknown origin) demethylation activity preincubated for 10 mins followed by peptide...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
Displayed 1 to 50 (of 143 total ) | Next | Last >>
Jump to: