Compile Data Set for Download or QSAR
Found 223 with Last Name = 'carbain' and Initial = 'b'
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235359(CHEMBL4088242)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235343(CHEMBL4103249)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235335(CHEMBL4092981)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235348(CHEMBL4078988)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235342(CHEMBL319467 | NU-6102)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235346(CHEMBL4102518)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235347(CHEMBL4078246)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553212(CHEMBL4763380)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553217(CHEMBL4761747)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233206(CHEMBL4059895)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C70PTPubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235349(CHEMBL4065402)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro inhibition against angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233212(CHEMBL4076762)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C70PTPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553207(CHEMBL4786783)copy SMILES
Affinity DataIC50: 18nMAssay Description:Inhibition of human NEK2 by kinase-profiling analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235336(CHEMBL4085238)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235354(CHEMBL4069161)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235344(CHEMBL4086832)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro inhibition against angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235345(CHEMBL4105278)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235340(CHEMBL4101626)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553200(CHEMBL4796125)copy SMILES
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235337(CHEMBL4062554)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233207(CHEMBL4098319)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C70PTPubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233211(CHEMBL4103466)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235355(CHEMBL4081027)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553205(CHEMBL4743876)copy SMILES
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553213(CHEMBL4779487)copy SMILES
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235334(CHEMBL4070391)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233213(CHEMBL4103343)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C70PTPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553201(CHEMBL4775990)copy SMILES
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetCyclin-A2(Bos taurus)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235356(CHEMBL4097571)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:In vitro inhibitory concentration against angiotensin-converting enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233966(CHEMBL4080296)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C70PTPubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233965(CHEMBL4093993)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C70PTPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553215(CHEMBL4783060)copy SMILES
Affinity DataIC50: 57nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553198(CHEMBL4796754)copy SMILES
Affinity DataIC50: 57nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553207(CHEMBL4786783)copy SMILES
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553204(CHEMBL4748191)copy SMILES
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50233967(CHEMBL4060905)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected insect Sf9 cells using histone H1 as substrate in presence of [gamma-3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C70PTPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553199(CHEMBL4795738)copy SMILES
Affinity DataIC50: 71nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553197(CHEMBL4746054)copy SMILES
Affinity DataIC50: 72nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553214(CHEMBL4776787)copy SMILES
Affinity DataIC50: 76nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553196(CHEMBL4783265)copy SMILES
Affinity DataIC50: 76nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553195(CHEMBL4746829)copy SMILES
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50553207(CHEMBL4786783)copy SMILES
Affinity DataIC50: 80nMAssay Description:Inhibition of Aurora A (unknown origin) preincubated with enzyme for 15 mins followed by substrate/ATP challenge for 90 mins by ProfilerPro plate bas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553209(CHEMBL4761123)copy SMILES
Affinity DataIC50: 88nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553208(CHEMBL4776060)copy SMILES
Affinity DataIC50: 93nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235343(CHEMBL4103249)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833V86PubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553210(CHEMBL4754015)copy SMILES
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553202(CHEMBL4753609)copy SMILES
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553203(CHEMBL4756141)copy SMILES
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))TBA
LigandPNGBDBM50553194(CHEMBL4759854)copy SMILES
Affinity DataIC50: 116nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50553207(CHEMBL4786783)copy SMILES
Affinity DataIC50: 120nMAssay Description:Inhibition of human NAUK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272RVPubMed
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