Compile Data Set for Download or QSAR
Found 371 with Last Name = 'grubinska' and Initial = 'b'
LigandPNGBDBM50341056(5-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3KbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341056(5-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of mTOR assessed as inhibition of phosphorylation of 4EBP1 by Lantha-Screen enzyme assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
LigandPNGBDBM50341056(5-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PI3KdeltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
LigandPNGBDBM50341056(5-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400752(CHEMBL2203552)copy SMILEScopy InChI
Affinity DataIC50: 1.49nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396302(CHEMBL2172485)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341035(1-(4-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-b...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of mTOR assessed as inhibition of phosphorylation of 4EBP1 by Lantha-Screen enzyme assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396298(CHEMBL2172489)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396305(CHEMBL2172482)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
LigandPNGBDBM50341054(3-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3KdeltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400756(CHEMBL2203562)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396301(CHEMBL2172486)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396316(CHEMBL2172635)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396297(CHEMBL2172490)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396322(CHEMBL2172629)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396308(CHEMBL2172636)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396307(CHEMBL2172480)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400754(CHEMBL2203564)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
LigandPNGBDBM50341054(3-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396303(CHEMBL2172484)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400753(CHEMBL2203565)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400757(CHEMBL2203561)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400755(CHEMBL2203563)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
LigandPNGBDBM50341056(5-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396299(CHEMBL2172488)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341056(5-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of mTOR in human U-87 cells assessed as inhibition of phosphorylation of AKT at S473More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396309(CHEMBL2172640)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396321(CHEMBL2172630)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
LigandPNGBDBM50341035(1-(4-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-b...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341054(3-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of mTOR assessed as inhibition of phosphorylation of 4EBP1 by Lantha-Screen enzyme assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
LigandPNGBDBM50341054(3-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341063(2-(4-(2-(3-hydroxyphenylamino)-1H-benzo[d]imidazol...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of mTOR assessed as inhibition of phosphorylation of 4EBP1 by Lantha-Screen enzyme assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400748(CHEMBL2203556)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400752(CHEMBL2203552)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396314(CHEMBL2172475)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400752(CHEMBL2203552)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of CK1-alpha using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 8 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341054(3-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of mTOR in human U-87 cells assessed as inhibition of phosphorylation of AKT at S473More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
LigandPNGBDBM50341054(3-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-benz...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of PI3KbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396300(CHEMBL2172487)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341035(1-(4-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-b...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of mTOR in human U-87 cells assessed as inhibition of phosphorylation of AKT at S473More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
LigandPNGBDBM50341035(1-(4-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-b...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of PI3KdeltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396312(CHEMBL2172637)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
LigandPNGBDBM50341035(1-(4-(1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-1H-b...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3KgammaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50341036(CHEMBL1760155 | N-(4-(1-(4-amino-6-methyl-1,3,5-tr...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of mTOR assessed as inhibition of phosphorylation of 4EBP1 by Lantha-Screen enzyme assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8MBWPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396326(CHEMBL2172625)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396296(CHEMBL2172477)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400751(CHEMBL2203553)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of CK1-delta using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 11 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396311(CHEMBL2172638)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400748(CHEMBL2203556)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Amgen Inc

Curated by ChEMBL
LigandPNGBDBM50396295(CHEMBL2172478)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of mTOR by LanthaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DHNPubMed
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