Compile Data Set for Download or QSAR
Found 197 with Last Name = 'klebl' and Initial = 'b'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50106301(CHEMBL3598140)copy SMILEScopy InChI
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595941(CHEMBL5200206)copy SMILES
Affinity DataIC50: 7.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595938(CHEMBL5197292)copy SMILES
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50106301(CHEMBL3598140)copy SMILEScopy InChI
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595941(CHEMBL5200206)copy SMILES
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595938(CHEMBL5197292)copy SMILES
Affinity DataIC50: 31nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595946(CHEMBL5180168)copy SMILES
Affinity DataIC50: 33nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168247(2,3-Di-thiophen-2-yl-benzo[g]quinoxaline-7-carboxy...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595945(CHEMBL5178739)copy SMILES
Affinity DataIC50: 46nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595944(CHEMBL5177875)copy SMILES
Affinity DataIC50: 74nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50519883(CHEMBL4522217)copy SMILEScopy InChI
Affinity DataIC50: 100nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595946(CHEMBL5180168)copy SMILES
Affinity DataIC50: 110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595945(CHEMBL5178739)copy SMILES
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595944(CHEMBL5177875)copy SMILES
Affinity DataIC50: 220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50519883(CHEMBL4522217)copy SMILEScopy InChI
Affinity DataIC50: 270nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595942(CHEMBL5177120)copy SMILES
Affinity DataIC50: 290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509371(CHEMBL4521241)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595942(CHEMBL5177120)copy SMILES
Affinity DataIC50: 490nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168248(CHEMBL192909 | {5-[3-(4-Carboxymethyl-thiophen-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 640nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168244(4-(5-{3-[5-(3-Carboxy-propyl)-thiophen-2-yl]-benzo...)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168242(3-(5-{3-[5-(2-Carboxy-ethyl)-thiophen-2-yl]-benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 870nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168241(6,7-Di-thiophen-2-yl-2,3-dihydro-1,4-dioxa-5,8-dia...)copy SMILEScopy InChI
Affinity DataIC50: 950nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168239(7,8-Dimethoxy-2,3-di-thiophen-2-yl-pyrazino[2,3-b]...)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168236(CHEMBL193162 | {5-[3-(5-Carboxymethyl-thiophen-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.28E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetRibosomal protein S6 kinase beta-2(Homo sapiens (Human))
Semmelweis University

Curated by ChEMBL
LigandPNGBDBM50168235(2,3-Di-thiophen-2-yl-benzo[g]quinoxaline | CHEMBL3...)copy SMILEScopy InChI
Affinity DataIC50: 1.36E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5'-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W37VVXPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595943(CHEMBL5189438)copy SMILES
Affinity DataIC50: 1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595948(CHEMBL5205628)copy SMILES
Affinity DataIC50: 1.80E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595947(CHEMBL5182239)copy SMILES
Affinity DataIC50: 1.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595939(CHEMBL5209370)copy SMILES
Affinity DataIC50: 2.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))TBA
LigandPNGBDBM50595948(CHEMBL5205628)copy SMILES
Affinity DataIC50: 2.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66QS1PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
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