Compile Data Set for Download or QSAR
Found 265 with Last Name = 'klenke' and Initial = 'b'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35836(pyrimidine-4-carboxamide, 118)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35834(pyrimidine-4-carboxamide, 116)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35829(pyrimidine-4-carboxamide, 111)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35833(pyrimidine-4-carboxamide, 115)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35784(pyrimidine-4-carboxamide, 19 | pyrimidine-4-carbox...)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35784(pyrimidine-4-carboxamide, 19 | pyrimidine-4-carbox...)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35843(pyrimidine-4-carboxamide, 28)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35830(pyrimidine-4-carboxamide, 112)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35832(pyrimidine-4-carboxamide, 114)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35837(pyrimidine-4-carboxamide, 119)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35786(pyrimidine-4-carboxamide, 27)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35785(pyrimidine-4-carboxamide, 25)copy SMILEScopy InChI
Affinity DataKi:  4.30nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35774(triazine-4-carboxamide, 6)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35835(pyrimidine-4-carboxamide, 117)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35839(pyrimidine-4-carboxamide, 121)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35845(pyrimidine-4-carboxamide, 58)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35838(pyrimidine-4-carboxamide, 120)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35841(pyrimidine-4-carboxamide, 123)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35777(triazine-4-carboxamide, 9)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35776(triazine-4-carboxamide, 8)copy SMILEScopy InChI
Affinity DataKi:  7.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35840(pyrimidine-4-carboxamide, 122)copy SMILEScopy InChI
Affinity DataKi:  8.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35782(triazine-4-carboxamide, 14)copy SMILEScopy InChI
Affinity DataKi:  8.80nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35810(pyrimidine-4-carboxamide, 70)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35806(pyrimidine-4-carboxamide, 62)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35831(pyrimidine-4-carboxamide, 113)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35820(pyrimidine-4-carboxamide, 91)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35775(triazine-4-carboxamide, 7)copy SMILEScopy InChI
Affinity DataKi:  12.3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35805(pyrimidine-4-carboxamide, 60)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35788(pyrimidine-4-carboxamide, 57)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35811(pyrimidine-4-carboxamide, 72)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35789(pyrimidine-4-carboxamide, 59)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35794(pyrimidine-4-carboxamide, 69)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35790(pyrimidine-4-carboxamide, 61)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35781(triazine-4-carboxamide, 13)copy SMILEScopy InChI
Affinity DataKi:  18.6nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35808(pyrimidine-4-carboxamide, 66)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35807(pyrimidine-4-carboxamide, 64)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35813(pyrimidine-4-carboxamide, 76)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35778(triazine-4-carboxamide, 10)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35821(pyrimidine-4-carboxamide, 93)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35797(pyrimidine-4-carboxamide, 75)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35809(pyrimidine-4-carboxamide, 68)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35818(pyrimidine-4-carboxamide, 86)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35812(pyrimidine-4-carboxamide, 74)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35791(pyrimidine-4-carboxamide, 63)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35806(pyrimidine-4-carboxamide, 62)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35792(pyrimidine-4-carboxamide, 65)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35795(pyrimidine-4-carboxamide, 71)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35790(pyrimidine-4-carboxamide, 61)copy SMILEScopy InChI
Affinity DataKi:  38nM ΔG°:  -41.8kJ/molepH: 7.5 T: 2°CAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35805(pyrimidine-4-carboxamide, 60)copy SMILEScopy InChI
Affinity DataKi:  38nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Vernalis (R&D) Ltd

LigandPNGBDBM35845(pyrimidine-4-carboxamide, 58)copy SMILEScopy InChI
Affinity DataKi:  38nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M069HPubMed
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