Compile Data Set for Download or QSAR
Found 130 with Last Name = 'lefranc' and Initial = 'b'
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347818(CHEMBL1802413 | P518)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469449(CHEMBL4277047)copy SMILEScopy InChI
Affinity DataIC50: 579nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396422(CHEMBL2170403)copy SMILEScopy InChI
Affinity DataIC50: 1.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)copy SMILEScopy InChI
Affinity DataIC50: 2.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469440(CHEMBL4281854)copy SMILEScopy InChI
Affinity DataIC50: 6.06E+3nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469430(CHEMBL4279100)copy SMILEScopy InChI
Affinity DataIC50: 8.25E+3nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347830(CHEMBL1802425)copy SMILEScopy InChI
Affinity DataIC50: 8.73E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396416(CHEMBL2170398)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396417(CHEMBL2170395)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396418(CHEMBL2170394)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396419(CHEMBL2170393)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as inhibition of human 26RFa-induced increase in intracell...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469444(CHEMBL4284790)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469445(CHEMBL4294578)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469431(CHEMBL4282568)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469447(CHEMBL4291594)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469448(CHEMBL4286672)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469451(CHEMBL4289785)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469424(CHEMBL4288232)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469452(CHEMBL4282993)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469432(CHEMBL4277540)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469435(CHEMBL4289249)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469438(CHEMBL4285426)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469426(CHEMBL4292045)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469433(CHEMBL4288190)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469443(CHEMBL4280959)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469441(CHEMBL4286363)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469428(CHEMBL4290858)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469427(CHEMBL4289720)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469420(CHEMBL4288630)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469421(CHEMBL4287681)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469422(CHEMBL4293167)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469437(CHEMBL4277480)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469429(CHEMBL4294254)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469442(CHEMBL4277203)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469434(CHEMBL4292662)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347858(CHEMBL1802423)copy SMILEScopy InChI
Affinity DataEC50:  233nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50469446(CHEMBL4288785)copy SMILEScopy InChI
Affinity DataEC50:  2.75E+3nMAssay Description:Agonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as increase Ca2+ mobilization after 3 mins by Fluo-4 AM-based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222XG4PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396422(CHEMBL2170403)copy SMILEScopy InChI
Affinity DataEC50:  94nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)copy SMILEScopy InChI
Affinity DataEC50:  136nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50396416(CHEMBL2170398)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35VSGPubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347818(CHEMBL1802413 | P518)copy SMILEScopy InChI
Affinity DataEC50:  10.4nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347819(CHEMBL1802414 | P550)copy SMILEScopy InChI
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347820(CHEMBL1802415)copy SMILEScopy InChI
Affinity DataEC50:  2.91E+3nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347821(CHEMBL1800099)copy SMILEScopy InChI
Affinity DataEC50:  43.2nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347822(CHEMBL1802418)copy SMILEScopy InChI
Affinity DataEC50:  30.2nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347823(CHEMBL1802419)copy SMILEScopy InChI
Affinity DataEC50:  37.5nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347824(CHEMBL1802420)copy SMILEScopy InChI
Affinity DataEC50:  95.3nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347825(CHEMBL1802417)copy SMILEScopy InChI
Affinity DataEC50:  185nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347826(CHEMBL1802416)copy SMILEScopy InChI
Affinity DataEC50:  138nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL
LigandPNGBDBM50347827(CHEMBL1802421)copy SMILEScopy InChI
Affinity DataEC50:  237nMAssay Description:Agonist activity at DYKDDDDK-flagged human GPR103 receptor expressed in CHO-K1 cells co-expressing G-protein alpha16 assessed as stimulation of calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40VJ8PubMed
Displayed 1 to 50 (of 130 total ) | Next | Last >>
Jump to: