Compile Data Set for Download or QSAR
Found 252 with Last Name = 'madeira' and Initial = 'b'
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073585(CHEMBL3408945 | US10358436, Example A102 | US99078...)copy SMILES
Affinity DataKi:  0.100nMAssay Description:Competitive binding to PLK4 (unknown origin) by double reciprocal plot analysis in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073587(CHEMBL3408947 | US10358436, Example A185 | US20230...)copy SMILES
Affinity DataKi:  0.260nMAssay Description:Competitive binding to PLK4 (unknown origin) by double reciprocal plot analysis in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081537(CHEMBL3422092)copy SMILES
Affinity DataKi:  0.700nMAssay Description:Competitive inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate by Lineweaver-Burk plot analysis in prese...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073586(CHEMBL3408946 | US10358436, Example A198 | US99078...)copy SMILES
Affinity DataKi:  0.730nMAssay Description:Competitive binding to PLK4 (unknown origin) by double reciprocal plot analysis in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183019(CHEMBL3819210)copy SMILEScopy InChI
Affinity DataKi:  0.770nMAssay Description:Competitive inhibition of TTK (unknown origin) by double reciprocal plot analysis in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044656(CHEMBL3353348 | US10358436, Example A35 | US990780...)copy SMILES
Affinity DataIC50: 0.370nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073551(CHEMBL3408955)copy SMILEScopy InChI
Affinity DataIC50: 0.390nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183021(CHEMBL3818646)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073584(CHEMBL3408944 | US10358436, Example A59 | US990780...)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073550(CHEMBL3408954)copy SMILEScopy InChI
Affinity DataIC50: 0.640nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183022(CHEMBL3819019)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044665(CHEMBL3353341 | US10358436, Example A33 | US990780...)copy SMILES
Affinity DataIC50: 0.75nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073555(CHEMBL3408941 | US10358436, Example A92 | US990780...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044662(CHEMBL3353361 | US10358436, Example A61 | US990780...)copy SMILES
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044667(CHEMBL3353362 | US10358436, Example A58 | US990780...)copy SMILES
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183023(CHEMBL3819328)copy SMILEScopy InChI
Affinity DataIC50: 0.940nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081539(CHEMBL3422104)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged TTK using biotinylated PWDPDDADITEILG as substrate preincubated for 15 mins followe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081539(CHEMBL3422104)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human TTKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073552(CHEMBL3408956 | US10358436, Example A78 | US990780...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081607(CHEMBL3422080)copy SMILES
Affinity DataIC50: 1.10nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081597(CHEMBL3422095)copy SMILES
Affinity DataIC50: 1.10nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044657(CHEMBL3353347 | US10358436, Example A24 | US990780...)copy SMILES
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044657(CHEMBL3353347 | US10358436, Example A24 | US990780...)copy SMILES
Affinity DataIC50: 1.10nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081578(CHEMBL3422091)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081578(CHEMBL3422091)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081574(CHEMBL3422086)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073554(CHEMBL3408940 | US10358436, Example A110 | US99078...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073585(CHEMBL3408945 | US10358436, Example A102 | US99078...)copy SMILES
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081609(CHEMBL3422084)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044675(CHEMBL3353354 | US10358436, Example A56 | US990780...)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183019(CHEMBL3819210)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073582(CHEMBL3408942 | US10358436, Example A109 | US99078...)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073547(CHEMBL3408951)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081600(CHEMBL3422099)copy SMILES
Affinity DataIC50: 1.5nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073553(CHEMBL3408957)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183036(CHEMBL3818403)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081598(CHEMBL3422097)copy SMILES
Affinity DataIC50: 1.70nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50073549(CHEMBL3408953 | US10358436, Example A72 | US990780...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081552(CHEMBL3422063)copy SMILES
Affinity DataIC50: 1.90nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081571(CHEMBL3422083)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081573(CHEMBL3422085)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044674(CHEMBL3353355 | US10358436, Example A42 | US990780...)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081601(CHEMBL3422102)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50044674(CHEMBL3353355 | US10358436, Example A42 | US990780...)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PLK4 (unknown origin) by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M0475VPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183041(CHEMBL3819003)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183025(CHEMBL3818533)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081605(CHEMBL3422077)copy SMILES
Affinity DataIC50: 2.5nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50183027(CHEMBL3817905)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of TTK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8NNBPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081551(CHEMBL3422062)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
EntreMed Inc.

Curated by ChEMBL
LigandPNGBDBM50081599(CHEMBL3422098)copy SMILES
Affinity DataIC50: 2.70nMAssay Description:Inhibition of amino terminal GST-fused full length human TTK using His6-SUMO-TTK-N as substrate preincubated for 15 mins prior to ATP addition by ind...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52RCNPubMed
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