Affinity DataKi: 0.200nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: >150nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: >150nMAssay Description:Antagonist activity at human histamine H3 receptor by [35S]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 323nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Antagonist potency against human H3 receptor in GTPgamma[S]-AssayMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by linear fitting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.30E+4nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by linear fitting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.90E+4nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by linear fitting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibiton of [3H]-ketanserin binding to human 5-HT2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [125I]-aminopotentidine binding to human H2 histamine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibiton of [3H]-ketanserin binding to human 5-HT2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]-pyrilamine binding to human H1 histamine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibiton of [3H]-histamine binding to human H4 histamine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+5nMAssay Description:Inhibition of recombinant F7a using S-2288 as substrate after 15 mins by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of F10a using S-2288 as substrate after 15 mins by competitive binding assayMore data for this Ligand-Target Pair
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