Compile Data Set for Download or QSAR
Found 51 with Last Name = 'suh' and Initial = 'bc'
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataKi:  0.00230nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220995(CHEMBL77788)copy SMILEScopy InChI
Affinity DataKi:  0.0190nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221005(CHEMBL75684)copy SMILEScopy InChI
Affinity DataKi:  0.0420nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220998(CHEMBL76382)copy SMILEScopy InChI
Affinity DataKi:  0.0460nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221003(CHEMBL432348)copy SMILEScopy InChI
Affinity DataKi:  0.0690nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220997(CHEMBL78237)copy SMILEScopy InChI
Affinity DataKi:  0.0920nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221006(CHEMBL77358)copy SMILEScopy InChI
Affinity DataKi:  0.146nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220999(CHEMBL77745)copy SMILEScopy InChI
Affinity DataKi:  0.336nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220996(CHEMBL76635)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221004(CHEMBL77999)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221001(CHEMBL76257)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220993(CHEMBL78238)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221007(CHEMBL80258)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221002(CHEMBL306320)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220994(CHEMBL77177)copy SMILEScopy InChI
Affinity DataKi: >5nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221000(CHEMBL431962)copy SMILEScopy InChI
Affinity DataKi: >5nMAssay Description:Binding affinity towards rolipram binding site on phosphodiesterase 4 using [3H]rolipram as radioligand in crude rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220996(CHEMBL76635)copy SMILEScopy InChI
Affinity DataIC50: 0.580nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221003(CHEMBL432348)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
The University of Texas

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]1,25-dihydroxyvitamin D3 from human VDR by HAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9QS7PubMedDrugBank
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220998(CHEMBL76382)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220993(CHEMBL78238)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221004(CHEMBL77999)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220995(CHEMBL77788)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036307(CHEMBL3353069)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036309(CHEMBL3353072)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221001(CHEMBL76257)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220999(CHEMBL77745)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036311(CHEMBL3353074)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221000(CHEMBL431962)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221006(CHEMBL77358)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50220994(CHEMBL77177)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221005(CHEMBL75684)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4C(Rattus norvegicus)
LEAD GENE CO., LTD

Curated by ChEMBL
LigandPNGBDBM50221002(CHEMBL306320)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against purified rat liver phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CZ39CGPubMed
TargetInositol 1,4,5-trisphosphate receptor type 3(Bos taurus)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50069314(CHEMBL346769 | D-MYO-INOSITOL 1,2,4,5-TETRAKISPHOS...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Binding affinity towards Inositol 1,4,5-trisphosphate receptor was evaluated by the standard competitive binding assay using 1.25 nM [3H]-D-I(1,4,5)P...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28051SQPubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50017691(CHEMBL126075 | dilazep)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036308(CHEMBL3353071)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
The University of Texas

Curated by ChEMBL
LigandPNGBDBM50200180(CHEMBL376093 | KSP-BCS-1-alpha-CHF2-20-epi-22-oxab...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]1,25-dihydroxyvitamin D3 from human VDR by HAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9QS7PubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
The University of Texas

Curated by ChEMBL
LigandPNGBDBM50200179((1S,3S,Z)-3-(difluoromethyl)-5-((E)-2-((1R,3aS,7aR...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]1,25-dihydroxyvitamin D3 from human VDR by HAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9QS7PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036310(CHEMBL3353073)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
The University of Texas

Curated by ChEMBL
LigandPNGBDBM50200181(CHEMBL220140 | KSP-BCS-1-alpha-CHF2-1624F2-2)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]1,25-dihydroxyvitamin D3 from human VDR by HAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9QS7PubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036306(CHEMBL3353070)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036314(CHEMBL3353077)copy SMILEScopy InChI
Affinity DataIC50: 94nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036313(CHEMBL3353076)copy SMILEScopy InChI
Affinity DataIC50: 217nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetInositol 1,4,5-trisphosphate receptor type 3(Bos taurus)
Pohang University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50069313(CHEMBL158474 | Phosphoric acid mono-((1S,2S,3R,4S,...)copy SMILEScopy InChI
Affinity DataIC50: 598nMAssay Description:Binding affinity towards Inositol 1,4,5-trisphosphate receptor was evaluated by the standard competitive binding assay using 1.25 nM [3H]-D-I(1,4,5)P...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28051SQPubMed
TargetEquilibrative nucleoside transporter 1(Homo sapiens (Human))
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036312(CHEMBL3353075)copy SMILEScopy InChI
Affinity DataIC50: 803nMAssay Description:Inhibition of human ENT1 expressed in porcine PK15NTD cells by cell-based [3H]5-uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetEquilibrative nucleoside transporter 2(Rattus norvegicus)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036307(CHEMBL3353069)copy SMILEScopy InChI
Affinity DataIC50: 977nMAssay Description:Inhibition of rat ENT2 expressed in rat H9c2 cells by cell-based 3H[5-]uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetEquilibrative nucleoside transporter 2(Rattus norvegicus)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036308(CHEMBL3353071)copy SMILEScopy InChI
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of rat ENT2 expressed in rat H9c2 cells by cell-based 3H[5-]uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetEquilibrative nucleoside transporter 2(Rattus norvegicus)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036306(CHEMBL3353070)copy SMILEScopy InChI
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of rat ENT2 expressed in rat H9c2 cells by cell-based 3H[5-]uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
TargetEquilibrative nucleoside transporter 2(Rattus norvegicus)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50036309(CHEMBL3353072)copy SMILEScopy InChI
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of rat ENT2 expressed in rat H9c2 cells by cell-based 3H[5-]uridine uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M38FZPubMed
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