Compile Data Set for Download or QSAR
Found 190 with Last Name = 'haug' and Initial = 'be'
TargetMyeloblastin(Homo sapiens (Human))
University of Bergen

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ349FPubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
UiT The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50166106(CHEMBL436283 | N-{3-[(2S,5S,8S,14R)-5-(3-Guanidino...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9SVZPubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
UiT The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50166087(CHEMBL436097 | N-{3-[(2R,5S,8S,14R)-5-(3-Guanidino...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9SVZPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509371(CHEMBL4521241)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMyeloblastin(Homo sapiens (Human))
University of Bergen

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ349FPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
UiT The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50100598(CHEMBL2031844)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9SVZPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 7(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GCK (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMyeloblastin(Homo sapiens (Human))
University of Bergen

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)copy SMILEScopy InChI
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ349FPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))TBA
LigandPNGBDBM50614333(CHEMBL5267172)copy SMILES
Affinity DataIC50: 7.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAurora kinase B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)copy SMILEScopy InChI
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of Aurora B (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))TBA
LigandPNGBDBM50614333(CHEMBL5267172)copy SMILES
Affinity DataIC50: 7.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of DRAK2 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))TBA
LigandPNGBDBM50614333(CHEMBL5267172)copy SMILES
Affinity DataIC50: 8.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCytochrome P450 2C9(Homo sapiens (Human))TBA
LigandPNGBDBM50614333(CHEMBL5267172)copy SMILES
Affinity DataIC50: 8.80E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50614333(CHEMBL5267172)copy SMILES
Affinity DataIC50: 9.30E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK2 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509369(CHEMBL4548361)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase SIK3(Homo sapiens)
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SIK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 11(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MLK3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of RIPK2 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509369(CHEMBL4548361)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetAurora kinase A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Aurora A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase 15(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509367(CHEMBL4476426)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ERK8 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509370(CHEMBL4446434)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK1A (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509368(CHEMBL4475097)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
TargetMitogen-activated protein kinase kinase kinase 9(Homo sapiens (Human))
UiT - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509366(CHEMBL4555884)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of MLK1 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M3B4RPubMed
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