Compile Data Set for Download or QSAR
Found 118 with Last Name = 'park' and Initial = 'bs'
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of ROS1 by HotSpot assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89CG9PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222640(CHEMBL415543)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222640(CHEMBL415543)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Korea University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of c-Met kinase (unknown origin)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222695(CHEMBL155433)copy SMILEScopy InChI
Affinity DataIC50: 0.460nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222637(CHEMBL154743)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222696(CHEMBL156041)copy SMILEScopy InChI
Affinity DataIC50: 0.550nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50296896((S)-2-(3-(3-hydroxy-5-methylphenyl)-4-(6-(2-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of ALK (unknown origin) incubated for 20 mins followed by [33P]ATP addition measured after 120 mins by HotSpot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50062357(AP26113 | CHEMBL3397300)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:Inhibition of ALK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of ROS1 (unknown origin)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222635(CHEMBL267205)copy SMILEScopy InChI
Affinity DataIC50: 0.720nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222647(CHEMBL154990)copy SMILEScopy InChI
Affinity DataIC50: 0.950nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222649(CHEMBL155730)copy SMILEScopy InChI
Affinity DataIC50: 0.950nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222641(CHEMBL157962)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50296896((S)-2-(3-(3-hydroxy-5-methylphenyl)-4-(6-(2-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of ROS1 (unknown origin) incubated for 20 mins followed by [33P]ATP addition measured after 120 mins by HotSpot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50062357(AP26113 | CHEMBL3397300)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of ROS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM482158(BDBM50242742 | TAE684)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of ROS1 (unknown origin) expressed in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222638(CHEMBL422702)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222644(CHEMBL434295)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM482158(BDBM50242742 | TAE684)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of ALK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222648(CHEMBL156693)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222639(CHEMBL356682)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222646(CHEMBL157917)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222694(CHEMBL158189)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222691(CHEMBL156927)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222690(CHEMBL345157)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of ROS1 (unknown origin) expressed in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Korea University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of c-Met kinase (unknown origin)More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Korea University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50296896((S)-2-(3-(3-hydroxy-5-methylphenyl)-4-(6-(2-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of c-Met (unknown origin) incubated for 20 mins followed by [33P]ATP addition measured after 120 mins by HotSpot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222645(CHEMBL157918)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222693(CHEMBL157579)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048844(CHEMBL3310332)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50062373(CHEMBL3397291)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of ROS1 (unknown origin) incubated for 20 mins followed by [33P]ATP addition measured after 120 mins by HotSpot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Korea University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of ALK (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048850(CHEMBL3310338)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222634(CHEMBL157473)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222643(CHEMBL157688)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222692(CHEMBL348634)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonistic activity against vanilloid receptor as concentration to reduce the response to 0.5 mM capsaicin by 50% from neonatal rat culture spinal ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP7747PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50062380(CHEMBL3397286)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of ROS1 (unknown origin) incubated for 20 mins followed by [33P]ATP addition measured after 120 mins by HotSpot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048849(CHEMBL3310337)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048857(CHEMBL3310324)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048854(CHEMBL3310326)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048841(CHEMBL3310329)copy SMILEScopy InChI
Affinity DataIC50: 74nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048845(CHEMBL3310333)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50062367(CHEMBL3397288)copy SMILEScopy InChI
Affinity DataIC50: 88nMAssay Description:Inhibition of ROS1 (unknown origin) incubated for 20 mins followed by [33P]ATP addition measured after 120 mins by HotSpot assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61MX6PubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048848(CHEMBL3310336)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048852(CHEMBL3310328)copy SMILEScopy InChI
Affinity DataIC50: 104nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048847(CHEMBL3310335)copy SMILEScopy InChI
Affinity DataIC50: 105nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50048856(CHEMBL3310325)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Inhibition of ROS1 (unknown origin) assessed as remaining activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765H0ZPubMed
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