TargetCyclin-G-associated kinase(Homo sapiens (Human))
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of tracer K5 binding to NanoLuc-fused CASK (unknown origin) expressed in HEK293T cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Binding affinity human SLK by binding displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Binding affinity human STK10 by binding displacement assayMore data for this Ligand-Target Pair