TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 26.7nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 111nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 196nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 207nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 223nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 291nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 315nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 383nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 540nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 737nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 827nMAssay Description:Binding affinity for recombinant rat alpha2-beta2-gamma2 GABA-A receptor subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 927nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 9.20E+4nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Universit£ degli Studi di Roma La Sapienza
Curated by ChEMBL
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of human recombinant GST-PRMT1 expressed in BL21 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of Aspergillus nidulans recombinant GST-RmtA expressed in BL21 cellsMore data for this Ligand-Target Pair