TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-Ro-15-1788 from rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]-Ro-15-1788 from rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-Ro-15-1788 from rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 13.9nMAssay Description:Displacement of [3H]-Ro-15-1788 from rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-Ro-15-1788 from rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 26.7nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 26.7nMAssay Description:Displacement of [3H]-Ro-15-1788 from rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]-Ro-15-1788 from rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha1-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 66nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:The compound was tested for its binding affinity towards Glycine/NMDA receptor in rat cortical membranes using [3H]-glycine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Inhibition by displacing [3H]-Glycine of N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 89nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity towards N-methyl-D-aspartate glutamate receptor 1 (high affinity) of rat cortical synaptic membranes by using [3H]-Gly as radioligan...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 111nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity towards N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranes using [3H]-glycine as radioligandMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 144nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha5/beta3/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 159nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha5/beta3/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Displacement of [3H]-Glycine from N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity towards N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranes using [3H]-glycine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition by displacing [3H]-Glycine of N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 196nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha3-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Ability of compound to displace [3H]-glycine from N-methyl-D-aspartate glutamate receptor 1 from in cerebral cortex synaptic membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 207nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2(Rattus norvegicus (Rat))
University of Firenze
Curated by ChEMBL
University of Firenze
Curated by ChEMBL
Affinity DataKi: 223nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha5-beta3-gamma2 subunits expresssed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement of [3H]-Glycine from N-methyl-D-aspartate glutamate receptor 1 in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Ability of compound to displace [3H]-glycine from N-methyl-D-aspartate glutamate receptor 1 from in cerebral cortex synaptic membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università degli Studi di Firenze
Curated by ChEMBL
Università degli Studi di Firenze
Curated by ChEMBL
Affinity DataKi: 285nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant rat GABAAalpha1/beta2/gamma2 receptor after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair