Compile Data Set for Download or QSAR
Found 153 with Last Name = 'el amri' and Initial = 'c'
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM588058(US11541023, Compound 6)copy SMILES
Affinity DataKi:  670nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM588055(US11541023, Compound 3)copy SMILES
Affinity DataKi:  790nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM50574434(CHEMBL4861066)copy SMILES
Affinity DataKi:  800nMAssay Description:Non-competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM588057(US11541023, Compound 5)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM50574435(CHEMBL4862261)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM50574434(CHEMBL4861066)copy SMILES
Affinity DataKi:  1.30E+3nMAssay Description:Competitive inhibition of plasmin (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM588055(US11541023, Compound 3)copy SMILES
Affinity DataKi:  1.32E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM50574432(CHEMBL4863108)copy SMILES
Affinity DataKi:  1.50E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM50574433(CHEMBL4852575)copy SMILES
Affinity DataKi:  1.50E+3nMAssay Description:Competitive inhibition of plasmin (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM588054(US11541023, Compound 2)copy SMILES
Affinity DataKi:  1.51E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM588058(US11541023, Compound 6)copy SMILES
Affinity DataKi:  1.75E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM588056(US11541023, Compound 4)copy SMILES
Affinity DataKi:  1.92E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM50574431(CHEMBL4847066)copy SMILES
Affinity DataKi:  2.00E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM588057(US11541023, Compound 5)copy SMILES
Affinity DataKi:  2.16E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM588054(US11541023, Compound 2)copy SMILES
Affinity DataKi:  2.26E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM50574433(CHEMBL4852575)copy SMILES
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetKallikrein-1(Homo sapiens (Human))TBA
LigandPNGBDBM50574434(CHEMBL4861066)copy SMILES
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of KLK1 (unknown origin) assessed as release of AMC fluorescent product using H-PFR-AMC as substrate incubated for 30 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM50574430(CHEMBL4853943)copy SMILES
Affinity DataKi:  4.30E+3nMAssay Description:Competitive inhibition of KLK6 (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)

Curated by ChEMBL
LigandPNGBDBM32709((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-met...)copy SMILEScopy InChI
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B61JVPubMed
TargetKallikrein-6(Homo sapiens (Human))TBA
LigandPNGBDBM588053(US11541023, Compound 1)copy SMILES
Affinity DataKi:  4.44E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM588056(US11541023, Compound 4)copy SMILES
Affinity DataKi:  4.66E+3nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM588053(US11541023, Compound 1)copy SMILES
Affinity DataKi:  1.44E+4nMAssay Description:In a typical test, 100 μl of reaction medium contains the buffer, 1 μl of recombinant enzyme, 1 μl of substrate (Boc-QAR-AMC) and 1 &#...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35ZH4US Patent
TargetPlasminogen(Homo sapiens (Human))TBA
LigandPNGBDBM50574430(CHEMBL4853943)copy SMILES
Affinity DataKi:  1.45E+4nMAssay Description:Competitive inhibition of plasmin (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89H6CPubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444601(CHEMBL3099881)copy SMILEScopy InChI
Affinity DataKi:  1.50E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50073221(CHEMBL3408420)copy SMILEScopy InChI
Affinity DataKi:  2.70E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P913VPubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444601(CHEMBL3099881)copy SMILEScopy InChI
Affinity DataKi:  4.40E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444600(CHEMBL1462676)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50073222(CHEMBL3125572)copy SMILEScopy InChI
Affinity DataKi:  5.06E+4nMAssay Description:Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P913VPubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444598(CHEMBL3099878)copy SMILEScopy InChI
Affinity DataKi:  5.50E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444604(CHEMBL3099870)copy SMILEScopy InChI
Affinity DataKi:  7.00E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444602(CHEMBL3099874)copy SMILEScopy InChI
Affinity DataKi:  7.20E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444603(CHEMBL3099871)copy SMILEScopy InChI
Affinity DataKi:  7.50E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444597(CHEMBL3099882)copy SMILEScopy InChI
Affinity DataKi:  8.30E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444599(CHEMBL3099875)copy SMILEScopy InChI
Affinity DataKi:  9.50E+4nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)

Curated by ChEMBL
LigandPNGBDBM50444597(CHEMBL3099882)copy SMILEScopy InChI
Affinity DataKi:  9.50E+4nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)

Curated by ChEMBL
LigandPNGBDBM50444602(CHEMBL3099874)copy SMILEScopy InChI
Affinity DataKi:  1.00E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)

Curated by ChEMBL
LigandPNGBDBM50444603(CHEMBL3099871)copy SMILEScopy InChI
Affinity DataKi:  1.07E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)

Curated by ChEMBL
LigandPNGBDBM50444604(CHEMBL3099870)copy SMILEScopy InChI
Affinity DataKi:  1.12E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)

Curated by ChEMBL
LigandPNGBDBM50444598(CHEMBL3099878)copy SMILEScopy InChI
Affinity DataKi:  1.21E+5nMAssay Description:Competitive inhibition of human kallikrein5 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444604(CHEMBL3099870)copy SMILEScopy InChI
Affinity DataKi:  1.29E+5nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444598(CHEMBL3099878)copy SMILEScopy InChI
Affinity DataKi:  1.31E+5nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444599(CHEMBL3099875)copy SMILEScopy InChI
Affinity DataKi:  1.40E+5nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444603(CHEMBL3099871)copy SMILEScopy InChI
Affinity DataKi:  1.52E+5nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444602(CHEMBL3099874)copy SMILEScopy InChI
Affinity DataKi:  1.64E+5nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444597(CHEMBL3099882)copy SMILEScopy InChI
Affinity DataKi:  1.66E+5nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM50444600(CHEMBL1462676)copy SMILEScopy InChI
Affinity DataKi:  1.66E+5nMAssay Description:Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21837Z8PubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM32709((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-met...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B61JVPubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universit£ Pierre et Marie Curie-Sorbonne Universit£s (UPMC)

Curated by ChEMBL
LigandPNGBDBM51911((4-isopropoxybenzyl)-[3-(2-methoxyphenyl)-3-(4-met...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B61JVPubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM33882((5-amino-3-pyridin-3-yl-1,2,4-triazol-1-yl)-(4-chl...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B61JVPubMed
TargetKallikrein-7(Homo sapiens (Human))
Universit£ Pierre et Marie Curie

Curated by ChEMBL
LigandPNGBDBM33437((5-amino-3-phenyl-1,2,4-triazol-1-yl)-(3,4-dimetho...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B61JVPubMed
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