Compile Data Set for Download or QSAR
Found 52 with Last Name = 'ferroud' and Initial = 'c'
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50525572(CH-223191 | CHEMBL1743245)copy SMILEScopy InChI
Affinity DataIC50: 2.43E+3nMAssay Description:Antagonist activity at AhR in human HepG2 cells assessed as inhibition of FICZ-induced AhR transcriptional activity incubated for 24 hrs by Quanti-Lu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239286(CHEMBL4084601)copy SMILEScopy InChI
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239287(CHEMBL4100095)copy SMILEScopy InChI
Affinity DataEC50:  6.80E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239288(CHEMBL4097685)copy SMILEScopy InChI
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239289(CHEMBL4096752)copy SMILEScopy InChI
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239290(CHEMBL4099197)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239291(CHEMBL4091463)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239284(CHEMBL4096360)copy SMILEScopy InChI
Affinity DataEC50:  4.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239285(CHEMBL4096869)copy SMILEScopy InChI
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239286(CHEMBL4084601)copy SMILEScopy InChI
Affinity DataEC50:  3.20E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239287(CHEMBL4100095)copy SMILEScopy InChI
Affinity DataEC50:  7.30E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239288(CHEMBL4097685)copy SMILEScopy InChI
Affinity DataEC50:  2.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239290(CHEMBL4099197)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+5nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239292(CHEMBL4070549)copy SMILEScopy InChI
Affinity DataEC50:  1.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239291(CHEMBL4091463)copy SMILEScopy InChI
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239293(CHEMBL4076088)copy SMILEScopy InChI
Affinity DataEC50:  1.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239294(CHEMBL4070517)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239292(CHEMBL4070549)copy SMILEScopy InChI
Affinity DataEC50:  1.90E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239293(CHEMBL4076088)copy SMILEScopy InChI
Affinity DataEC50:  3.00E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239289(CHEMBL4096752)copy SMILEScopy InChI
Affinity DataEC50:  2.70E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556458(CHEMBL4744715)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556459(CHEMBL4763780)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556460(CHEMBL4752532)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556461(CHEMBL4778652)copy SMILES
Affinity DataEC50: >4.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556462(CHEMBL4740412)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556463(CHEMBL4743405)copy SMILES
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556464(CHEMBL4789305)copy SMILES
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556465(CHEMBL4754940)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556466(CHEMBL4747237)copy SMILES
Affinity DataEC50: >2.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556467(CHEMBL4784860)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556468(CHEMBL4743891)copy SMILES
Affinity DataEC50: >2.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556469(CHEMBL4756557)copy SMILES
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556470(CHEMBL4760281)copy SMILES
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556471(CHEMBL4743041)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556472(CHEMBL4749793)copy SMILES
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556473(CHEMBL4746741)copy SMILES
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556474(CHEMBL4758967)copy SMILES
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556475(CHEMBL4764664)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556476(CHEMBL4796168)copy SMILES
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556477(CHEMBL4756836)copy SMILES
Affinity DataEC50:  5.36E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556478(CHEMBL4742377)copy SMILES
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556479(CHEMBL4757889)copy SMILES
Affinity DataEC50: >2.00E+5nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556480(CHEMBL4756642)copy SMILES
Affinity DataEC50:  2.17E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556481(CHEMBL4747529)copy SMILES
Affinity DataEC50:  2.79E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556482(CHEMBL4758893)copy SMILES
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556483(CHEMBL4749256)copy SMILES
Affinity DataEC50:  1.32E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556484(CHEMBL4760226)copy SMILES
Affinity DataEC50:  1.99E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50556485(CHEMBL4798147)copy SMILES
Affinity DataEC50:  5.20E+4nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM61400(BISACODYL | MLS000069729 | SMR000058226 | cid_2391)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at AhR in human HepG2 cells co-transfected with pSELECT-zeo-Lucia and CYP1A1 assessed as induction of receptor transactivation incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
TargetAryl hydrocarbon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50541262(6-Formylindolo[3,2-B]Carbazole | CHEMBL472031)copy SMILEScopy InChI
Affinity DataEC50:  9.06E+3nMAssay Description:Agonist activity at AhR in human HepG2 cells assessed as induction of AhR transcriptional activity incubated for 24 hrs by Quanti-Luc reagent based l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P359JPubMed
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