Compile Data Set for Download or QSAR
Found 53 with Last Name = 'finamore' and Initial = 'c'
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535422(CHEMBL4527193)copy SMILEScopy InChI
Affinity DataIC50: 127nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535427(CHEMBL4464270)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535416(CHEMBL4451559)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+3nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535421(CHEMBL4519624)copy SMILEScopy InChI
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535420(CHEMBL4541043)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535425(CHEMBL4562404)copy SMILEScopy InChI
Affinity DataIC50: 2.05E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535417(CHEMBL4575954)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535423(CHEMBL4573467)copy SMILEScopy InChI
Affinity DataIC50: 2.57E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535426(CHEMBL4539531)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535419(CHEMBL4464005)copy SMILEScopy InChI
Affinity DataIC50: 2.84E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535418(CHEMBL4457628)copy SMILEScopy InChI
Affinity DataIC50: 3.38E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535428(CHEMBL4452655)copy SMILEScopy InChI
Affinity DataIC50: 3.45E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535424(CHEMBL4564891)copy SMILEScopy InChI
Affinity DataIC50: 4.04E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R07PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535376(CHEMBL4451432)copy SMILEScopy InChI
Affinity DataEC50:  1.59E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM21724(3-[(E)-2-(2-chloro-4-{[3-(2,6-dichlorophenyl)-5-(1...)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM21675((4R)-4-[(1S,2S,5R,7S,8R,9R,10S,11S,14R,15R)-8-ethy...)copy SMILEScopy InChI
Affinity DataEC50:  500nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535377(CHEMBL4553281)copy SMILEScopy InChI
Affinity DataEC50:  740nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535378(CHEMBL4562865)copy SMILEScopy InChI
Affinity DataEC50:  2.80E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535379(CHEMBL4445722)copy SMILEScopy InChI
Affinity DataEC50:  1.40E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535380(CHEMBL4578551)copy SMILEScopy InChI
Affinity DataEC50:  5.40E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535381(CHEMBL4591419)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535382(CHEMBL4588863)copy SMILEScopy InChI
Affinity DataEC50:  460nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535383(CHEMBL4436469)copy SMILEScopy InChI
Affinity DataEC50:  2.93E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM21674((4R)-4-[(1S,2S,5R,7S,9R,10R,11S,14R,15R)-5,9-dihyd...)copy SMILEScopy InChI
Affinity DataEC50:  2.00E+4nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535384(CHEMBL4465344)copy SMILEScopy InChI
Affinity DataEC50:  1.97E+4nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535385(CHEMBL4455475)copy SMILEScopy InChI
Affinity DataEC50:  670nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535386(CHEMBL4535914)copy SMILEScopy InChI
Affinity DataEC50:  3.59E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535387(CHEMBL4585144)copy SMILEScopy InChI
Affinity DataEC50:  830nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540717(CHEMBL4643260)copy SMILEScopy InChI
Affinity DataEC50:  2.65E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540718(CHEMBL4635684)copy SMILEScopy InChI
Affinity DataEC50:  6.90E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540719(CHEMBL4643368)copy SMILEScopy InChI
Affinity DataEC50:  570nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540720(CHEMBL4647613)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540721(CHEMBL4646200)copy SMILEScopy InChI
Affinity DataEC50:  660nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540722(CHEMBL4648823)copy SMILEScopy InChI
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540723(CHEMBL4638053)copy SMILEScopy InChI
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540724(CHEMBL4646264)copy SMILEScopy InChI
Affinity DataEC50:  2.26E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540725(CHEMBL4637054)copy SMILEScopy InChI
Affinity DataEC50:  780nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540726(CHEMBL4635505)copy SMILEScopy InChI
Affinity DataEC50:  4.58E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50540727(CHEMBL4642126)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PD0PubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535375(CHEMBL4592387)copy SMILEScopy InChI
Affinity DataEC50:  6.67E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535374(CHEMBL4591348)copy SMILEScopy InChI
Affinity DataEC50:  2.06E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535373(CHEMBL4471591)copy SMILEScopy InChI
Affinity DataEC50:  1.02E+4nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535372(CHEMBL4532035)copy SMILEScopy InChI
Affinity DataEC50:  1.15E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535371(CHEMBL4455911)copy SMILEScopy InChI
Affinity DataEC50:  730nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535370(CHEMBL4448603)copy SMILEScopy InChI
Affinity DataEC50:  810nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535369(CHEMBL4461163)copy SMILEScopy InChI
Affinity DataEC50:  940nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535368(CHEMBL4450943)copy SMILEScopy InChI
Affinity DataEC50:  4.37E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetBile acid receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50535367(CHEMBL4456883)copy SMILEScopy InChI
Affinity DataEC50:  1.09E+3nMAssay Description:Transactivation of human FXR (unknown origin) expressed in HepG2 cells co-expressing pSG5RXR/pGL4.70 after 24 hrs post transfection by luciferase rep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1HXKPubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50028027(CHEMBL3342086)copy SMILEScopy InChI
Affinity DataEC50:  400nMAssay Description:Agonist activity at GP-BAR1 (unknown origin) in human HEK293 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs by CR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5WMNPubMed
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50028028(CHEMBL3342082)copy SMILEScopy InChI
Affinity DataEC50:  1.03E+3nMAssay Description:Agonist activity at GP-BAR1 (unknown origin) in human HEK293 cells assessed as receptor transactivation at 100 nM to 50 uM incubated for 16 hrs by CR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5WMNPubMed
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