TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Bcl-xL/BAK (unknown origin) interactionMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of Bcl-xL/BAK (unknown origin) interactionMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of Bcl-xL/BAK (unknown origin) interactionMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of Bcl-xL/BAK (unknown origin) interactionMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of Bcl-xL/BAK (unknown origin) interactionMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 115nMAssay Description:Inhibition of Bcl-xL/BAK (unknown origin) interactionMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 142nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of MCL1 binding to Bak by FRET assayMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of Bcl-2/biotinylated BAK (unknown origin) interaction incubated for 1 hr by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of human HDAC1 assessed as [3H]acetate release after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of Mcl1 protein by Mcl1/Bak fluorescence resonance assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of Mcl1 protein by Mcl1/Bak fluorescence resonance assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Harbor Branch Oceanographic Institute at Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of Bak binding to Mcl-1 by FRET assayMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 5nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 104nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 2nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 8nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 7nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 10nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 14nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 17nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 0.600nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Novartis Institutes for BioMedical Research Inc.
Curated by ChEMBL
Affinity DataKd: 3nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
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