Compile Data Set for Download or QSAR
Found 155 with Last Name = 'jenkinson' and Initial = 'c'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Research and Development LLC

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7K4TPubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268488(CHEMBL4092882)copy SMILEScopy InChI
Affinity DataEC50:  142nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268489(CHEMBL4065220)copy SMILEScopy InChI
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268490(CHEMBL4072480)copy SMILEScopy InChI
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268491(CHEMBL4073815)copy SMILEScopy InChI
Affinity DataEC50:  520nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268496(CHEMBL4062462)copy SMILEScopy InChI
Affinity DataEC50:  610nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268497(CHEMBL4084166)copy SMILEScopy InChI
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268498(CHEMBL4076902)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268499(CHEMBL4061340)copy SMILEScopy InChI
Affinity DataEC50:  145nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268503(CHEMBL4083233)copy SMILEScopy InChI
Affinity DataEC50:  220nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268491(CHEMBL4073815)copy SMILEScopy InChI
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268496(CHEMBL4062462)copy SMILEScopy InChI
Affinity DataEC50:  2.03E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268498(CHEMBL4076902)copy SMILEScopy InChI
Affinity DataEC50:  750nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268499(CHEMBL4061340)copy SMILEScopy InChI
Affinity DataEC50:  930nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268504(CHEMBL4070355)copy SMILEScopy InChI
Affinity DataEC50:  410nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268505(CHEMBL4083499)copy SMILEScopy InChI
Affinity DataEC50:  150nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268506(CHEMBL4061699)copy SMILEScopy InChI
Affinity DataEC50:  71nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268507(CHEMBL4073078)copy SMILEScopy InChI
Affinity DataEC50:  670nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268515(CHEMBL4099943)copy SMILEScopy InChI
Affinity DataEC50:  680nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268516(CHEMBL4084679)copy SMILEScopy InChI
Affinity DataEC50:  2.83E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268517(CHEMBL4063013)copy SMILEScopy InChI
Affinity DataEC50:  1.07E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268518(CHEMBL4074388)copy SMILEScopy InChI
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268519(CHEMBL4101135)copy SMILEScopy InChI
Affinity DataEC50:  740nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268520(CHEMBL4065769)copy SMILEScopy InChI
Affinity DataEC50:  350nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268521(CHEMBL4093383)copy SMILEScopy InChI
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268522(CHEMBL4103573)copy SMILEScopy InChI
Affinity DataEC50:  1.44E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268523(CHEMBL4085643)copy SMILEScopy InChI
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268515(CHEMBL4099943)copy SMILEScopy InChI
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268536(CHEMBL4099026)copy SMILEScopy InChI
Affinity DataEC50:  150nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268537(CHEMBL4080995)copy SMILEScopy InChI
Affinity DataEC50:  170nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268538(CHEMBL4091291)copy SMILEScopy InChI
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268506(CHEMBL4061699)copy SMILEScopy InChI
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268537(CHEMBL4080995)copy SMILEScopy InChI
Affinity DataEC50:  69nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268536(CHEMBL4099026)copy SMILEScopy InChI
Affinity DataEC50:  230nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268539(CHEMBL4060663)copy SMILEScopy InChI
Affinity DataEC50:  290nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268540(CHEMBL4104082)copy SMILEScopy InChI
Affinity DataEC50:  180nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268541(CHEMBL4086174)copy SMILEScopy InChI
Affinity DataEC50:  60nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268542(CHEMBL4078286)copy SMILEScopy InChI
Affinity DataEC50:  190nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268543(CHEMBL4067368)copy SMILEScopy InChI
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268544(CHEMBL4095819)copy SMILEScopy InChI
Affinity DataEC50:  190nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268545(CHEMBL4077787)copy SMILEScopy InChI
Affinity DataEC50:  217nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268546(CHEMBL4062742)copy SMILEScopy InChI
Affinity DataEC50:  81nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268551(CHEMBL4103081)copy SMILEScopy InChI
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux by Fluo-4 NW dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268488(CHEMBL4092882)copy SMILEScopy InChI
Affinity DataEC50:  711nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268551(CHEMBL4103081)copy SMILEScopy InChI
Affinity DataEC50:  900nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268545(CHEMBL4077787)copy SMILEScopy InChI
Affinity DataEC50:  1.34E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268522(CHEMBL4103573)copy SMILEScopy InChI
Affinity DataEC50:  2.76E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268521(CHEMBL4093383)copy SMILEScopy InChI
Affinity DataEC50:  760nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268520(CHEMBL4065769)copy SMILEScopy InChI
Affinity DataEC50:  810nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Cardiovascular and Metabolic Research, Janssen Research& Development, LLC, Welsh& McKean Roads, Box 776, Spring House, PA 19477, United States. Electronic address: xzhang5@its.jnj.com.

Curated by ChEMBL
LigandPNGBDBM50268519(CHEMBL4101135)copy SMILEScopy InChI
Affinity DataEC50:  400nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as increase in intracellular calcium flux by DiscoveRx PathHunter beta-arrestin a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85BK4PubMed
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