Compile Data Set for Download or QSAR
Found 85 with Last Name = 'martyr' and Initial = 'c'
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498523(CHEMBL3605643)copy SMILEScopy InChI
Affinity DataKi:  0.00150nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 (HIV-1))
Purdue Research Foundation

US Patent
LigandPNGBDBM128418(US8802724, 23a | US8802724, 23c)copy SMILEScopy InChI
Affinity DataKi:  0.00290nMAssay Description:The enzyme inhibitory activity (Ki) was determined according to an assay protocol reported by Toth and Marshall (Toth, M. V.; Marshall, G. R. Int. J....More data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498524(CHEMBL3605638)copy SMILEScopy InChI
Affinity DataKi:  0.00390nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50489369(CHEMBL1232930 | GRL-0519)copy SMILEScopy InChI
Affinity DataKi:  0.00600nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498534(CHEMBL3605635)copy SMILEScopy InChI
Affinity DataKi:  0.00630nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498528(CHEMBL3605644)copy SMILEScopy InChI
Affinity DataKi:  0.00990nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493304(CHEMBL2426453)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498531(CHEMBL3605642)copy SMILEScopy InChI
Affinity DataKi:  0.0120nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 (HIV-1))
Purdue Research Foundation

US Patent
LigandPNGBDBM128417(US8802724, 3a)copy SMILEScopy InChI
Affinity DataKi:  0.0140nMAssay Description:The enzyme inhibitory activity (Ki) was determined according to an assay protocol reported by Toth and Marshall (Toth, M. V.; Marshall, G. R. Int. J....More data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498530(CHEMBL3605637)copy SMILEScopy InChI
Affinity DataKi:  0.0140nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498526(CHEMBL3605636)copy SMILEScopy InChI
Affinity DataKi:  0.0140nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498527(CHEMBL3605640)copy SMILEScopy InChI
Affinity DataKi:  0.0140nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM8125((3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl N-[(2S...)copy SMILEScopy InChI
Affinity DataKi:  0.0160nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493301(CHEMBL2426458)copy SMILEScopy InChI
Affinity DataKi:  0.0210nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498532(CHEMBL3605641)copy SMILEScopy InChI
Affinity DataKi:  0.0240nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498533(CHEMBL3605646)copy SMILEScopy InChI
Affinity DataKi:  0.0270nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 (HIV-1))
Purdue Research Foundation

US Patent
LigandPNGBDBM128418(US8802724, 23a | US8802724, 23c)copy SMILEScopy InChI
Affinity DataKi:  0.0350nMAssay Description:The enzyme inhibitory activity (Ki) was determined according to an assay protocol reported by Toth and Marshall (Toth, M. V.; Marshall, G. R. Int. J....More data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498529(CHEMBL3605645)copy SMILEScopy InChI
Affinity DataKi:  0.0480nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 (HIV-1))
Purdue Research Foundation

US Patent
LigandPNGBDBM128419(US8802724, 23b | US8802724, 23d)copy SMILEScopy InChI
Affinity DataKi:  0.0730nMAssay Description:The enzyme inhibitory activity (Ki) was determined according to an assay protocol reported by Toth and Marshall (Toth, M. V.; Marshall, G. R. Int. J....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445K5DUS Patent
TargetGag-Pol polyprotein(Human immunodeficiency virus type 1 (HIV-1))
Purdue Research Foundation

US Patent
LigandPNGBDBM128419(US8802724, 23b | US8802724, 23d)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:The enzyme inhibitory activity (Ki) was determined according to an assay protocol reported by Toth and Marshall (Toth, M. V.; Marshall, G. R. Int. J....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445K5DUS Patent
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493306(CHEMBL2426457)copy SMILEScopy InChI
Affinity DataKi:  0.410nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493305(CHEMBL2426454)copy SMILEScopy InChI
Affinity DataKi:  0.450nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50498525(CHEMBL3605639)copy SMILEScopy InChI
Affinity DataKi:  0.530nMAssay Description:Inhibition of HIV1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862KFSPubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493303(CHEMBL2426451)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493302(CHEMBL2426450)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493300(CHEMBL2426455)copy SMILEScopy InChI
Affinity DataKi:  8.80nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493308(CHEMBL2426452)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50493307(CHEMBL2426456)copy SMILEScopy InChI
Affinity DataKi:  139nMAssay Description:Inhibition of HIV1 LAI protease by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K07764PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607602(CHEMBL5220994)copy SMILES
Affinity DataIC50: 0.0794nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607596(CHEMBL5221053)copy SMILES
Affinity DataIC50: 0.100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607597(CHEMBL5219157)copy SMILES
Affinity DataIC50: 0.126nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607595(CHEMBL5219030)copy SMILES
Affinity DataIC50: 0.158nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607593(CHEMBL5219693)copy SMILES
Affinity DataIC50: 0.158nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607601(CHEMBL5219667)copy SMILES
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607598(CHEMBL5220447)copy SMILES
Affinity DataIC50: 0.251nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607599(CHEMBL5220732)copy SMILES
Affinity DataIC50: 0.251nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607600(CHEMBL5220956)copy SMILES
Affinity DataIC50: 0.316nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607589(CHEMBL5219678)copy SMILES
Affinity DataIC50: 0.398nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607585(CHEMBL5219512)copy SMILES
Affinity DataIC50: 0.631nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607600(CHEMBL5220956)copy SMILES
Affinity DataIC50: 0.631nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607588(CHEMBL5220546)copy SMILES
Affinity DataIC50: 0.794nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607586(CHEMBL5221030)copy SMILES
Affinity DataIC50: 0.794nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607590(CHEMBL5220332)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607605(CHEMBL5219177)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607592(CHEMBL5219466)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607584(CHEMBL5221088)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607577(CHEMBL5219851)copy SMILES
Affinity DataIC50: 7.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607604(CHEMBL5219712)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607580(CHEMBL5218875)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))TBA
LigandPNGBDBM50607594(CHEMBL5219204)copy SMILES
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P93H2PubMed
Displayed 1 to 50 (of 85 total ) | Next | Last >>
Jump to: