Affinity DataKi: 0.0648nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0711nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0908nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0916nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0939nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0954nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0970nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.105nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.114nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.122nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.139nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.145nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.172nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.176nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.185nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.214nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.371nMAssay Description:Displacement of [3H]-nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human mu opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human kappa opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Centro de Investigaci�n Lilly
Curated by ChEMBL
Centro de Investigaci�n Lilly
Curated by ChEMBL
Affinity DataKi: >375nMAssay Description:Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assayMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Eli Lilly and Company
Curated by ChEMBL
Eli Lilly and Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant AKT1 expressed in insect cells incubated for 60 mins measured at apparent ATP Km level by kinase ADP-FP assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Eli Lilly and Company
Curated by ChEMBL
Eli Lilly and Company
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human p70S6K measured at apparent ATP Km levelMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Eli Lilly and Company
Curated by ChEMBL
Eli Lilly and Company
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant AKT1 expressed in insect cells incubated for 60 mins measured at apparent ATP Km level by kinase ADP-FP assayMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Eli Lilly and Company
Curated by ChEMBL
Eli Lilly and Company
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant AKT1 expressed in insect cells incubated for 60 mins measured at apparent ATP Km level by kinase ADP-FP assayMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Eli Lilly and Company
Curated by ChEMBL
Eli Lilly and Company
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant AKT1 expressed in insect cells incubated for 60 mins measured at apparent ATP Km level by kinase ADP-FP assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Eli Lilly and Company
Curated by ChEMBL
Eli Lilly and Company
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human RSK1 measured at apparent ATP Km levelMore data for this Ligand-Target Pair
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