Compile Data Set for Download or QSAR
Found 29 with Last Name = 'meere' and Initial = 'c'
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of IK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM31774(CHEMBL104 | Canesten | Clotrimazole | Lotrimin | M...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMedDrugBank
LigandPNGBDBM31774(CHEMBL104 | Canesten | Clotrimazole | Lotrimin | M...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of IK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMedDrugBank
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279024((1,3-dimethyl-1H-pyrazol-5-yl)(5-(furan-2-carbonyl...)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278971(2-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279105(5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279065(5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278972(CHEMBL500166 | methyl 2-(5-(furan-2-carbonyl)-5,6-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278973((5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278994(CHEMBL498728 | phenanthridine-5,6(6H)-diylbis(fura...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278938(1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279063(5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one | CHEMBL49...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279105(5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279066(5-(3-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279104(5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278939((6-(cyclobutanecarbonyl)phenanthridin-5(6H)-yl)(fu...)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278936(1-(6-(1H-indol-3-yl)phenanthridin-5(6H)-yl)ethanon...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279063(5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one | CHEMBL49...)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM31774(CHEMBL104 | Canesten | Clotrimazole | Lotrimin | M...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279065(5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50278937(1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)copy SMILEScopy InChI
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279064(5-(4-nitrophenylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4SC AG

Curated by ChEMBL
LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
LigandPNGBDBM50279104(5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed