Compile Data Set for Download or QSAR
Found 67 with Last Name = 'muller' and Initial = 'c'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465543(CHEMBL4278778)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465543(CHEMBL4278778)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465544(CHEMBL4285802)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465534(CHEMBL4288560)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465540(CHEMBL4282396)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465536(CHEMBL4282793)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465539(CHEMBL4292433)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465541(CHEMBL4284735)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465535(CHEMBL4278314)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465533(CHEMBL4289190)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465537(CHEMBL4286225)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465546(CHEMBL4277865)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465545(CHEMBL4293000)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465538(CHEMBL4284197)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465548(CHEMBL4286686)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465547(CHEMBL4292615)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465542(CHEMBL4281327)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465551(CHEMBL4290684)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465549(CHEMBL1721265)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465550(CHEMBL4289645)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Bos taurus)
Université Louis Pasteur

Curated by ChEMBL
LigandPNGBDBM50242771(8-Benzyl-2-methyl-4-(N-methylamino)pyrazolo[1,5-a]...)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+4nMAssay Description:Inhibition of bovine aorta PDE2 in presence of cGMPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76C9XPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465535(CHEMBL4278314)copy SMILEScopy InChI
Affinity DataKd:  560nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465536(CHEMBL4282793)copy SMILEScopy InChI
Affinity DataKd:  890nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465537(CHEMBL4286225)copy SMILEScopy InChI
Affinity DataKd:  590nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465538(CHEMBL4284197)copy SMILEScopy InChI
Affinity DataKd:  940nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465544(CHEMBL4285802)copy SMILEScopy InChI
Affinity DataKd:  360nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465545(CHEMBL4293000)copy SMILEScopy InChI
Affinity DataKd:  860nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465540(CHEMBL4282396)copy SMILEScopy InChI
Affinity DataKd:  310nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465533(CHEMBL4289190)copy SMILEScopy InChI
Affinity DataKd:  770nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465539(CHEMBL4292433)copy SMILEScopy InChI
Affinity DataKd:  320nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465543(CHEMBL4278778)copy SMILEScopy InChI
Affinity DataKd:  190nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465546(CHEMBL4277865)copy SMILEScopy InChI
Affinity DataKd:  540nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University

Curated by ChEMBL
LigandPNGBDBM50465541(CHEMBL4284735)copy SMILEScopy InChI
Affinity DataKd:  410nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52S95PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263760(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263741(US9714221, Example 75)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263723(6-(2- chlorophenyl)- 5-[4- [(3S)-1-(3- fluoropropy...)copy SMILEScopy InChI
Affinity DataEC50:  0.700nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263702(6-(3-chloro-2-fluoro-phenyl)-5-[4-[(3S)-1-(3-fluor...)copy SMILEScopy InChI
Affinity DataEC50:  0.5nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263671(6-(2- chloro-3- fluoro- phenyl)-5- [4-[(3S)-1- (3-...)copy SMILEScopy InChI
Affinity DataEC50:  0.5nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263674(US9714221, Example 11)copy SMILEScopy InChI
Affinity DataEC50:  0.700nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263664(US9714221, Example 1)copy SMILEScopy InChI
Affinity DataEC50:  0.400nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50505996(CHEMBL4533966 | US11149031, Example 2)copy SMILEScopy InChI
Affinity DataEC50:  0.300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50505997(CHEMBL4572640)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263850(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263913(6-(4- chloro- phenyl)-5-[4- [(3S)-1-(3- fluoroprop...)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263919(US9714221, Example 215)copy SMILES
Affinity DataEC50:  1.5nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263678(6-(4- chloro-2- fluoro- phenyl)-5- [4-[(3S)-1- (3-...)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263667(US9714221, Example 4)copy SMILEScopy InChI
Affinity DataEC50:  0.300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50505998(CHEMBL4563508)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263675(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)copy SMILES
Affinity DataEC50:  0.5nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM263681(6-(2,4- dichloro- phenyl)-5-[4- [(3S)-1-(3- fluoro...)copy SMILEScopy InChI
Affinity DataEC50:  0.900nMAssay Description:Induction of ERalpha degradation in human MCF7 cells incubated for 4 hrs by Alexafluor-488 conjugate anti-rabbit antibody/Syto-64 staining based immu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154MB3PubMed
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