Compile Data Set for Download or QSAR
Found 409 with Last Name = 'peifer' and Initial = 'c'
TargetProtein-serine O-palmitoleoyltransferase porcupine(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50133864(CHEMBL2139947 | US10251893, Compound 59)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of porcupine in HEK293T cells transfected with Wnt3A-expressing vector assessed as suppression of Wnt/beta-catenin signaling after 22 hrs ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4F5DPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM47167(CHEMBL201511 | US8957103, Z1 | US9364459, A)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FQSPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM47167(CHEMBL201511 | US8957103, Z1 | US9364459, A)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human VEGFR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8794PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM47167(CHEMBL201511 | US8957103, Z1 | US9364459, A)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human VEGFR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC108SPubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM47167(CHEMBL201511 | US8957103, Z1 | US9364459, A)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FQSPubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM47167(CHEMBL201511 | US8957103, Z1 | US9364459, A)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human VEGFR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8794PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300888((S)-4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen

Curated by ChEMBL
LigandPNGBDBM50516619(CHEMBL4547542)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2ZWXPubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...)copy SMILEScopy InChI
Affinity DataIC50: 9.60nMAssay Description:Inhibition of human recombinant BRAF V600E mutant using MEK1 as substrate measured after 1 hr by Western blot analysisMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetPyruvate kinase(Staphylococcus aureus (strain MRSA252))
Christian-Albrechts-University of Kiel

Curated by ChEMBL
LigandPNGBDBM50192869(CIS-3,4-DIHYDROHAMACANTHIN B)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of methicillin-resistant Staphylococcus aureus pyruvate kinase by coupled lactate dehydrogenase continuous assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Christian-Albrechts-University of Kiel

Curated by ChEMBL
LigandPNGBDBM50192877(CHEMBL3358999)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant PDGFRbeta using poly(Ala,Glu,Lys,Tyr) substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6V0RPubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen

Curated by ChEMBL
LigandPNGBDBM50484216(CHEMBL1822256)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant BRAF V600E mutant using MEK1 as substrate measured after 1 hr by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2ZWXPubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human CK1delta transcription variant 1 using GST-tagged mouse p53 (1 to 64 residues) as substrate in presence of radiolabelled-ATP by C...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300885(CHEMBL569551 | N-sec-butyl-4-(3-(4-fluorophenyl)-5...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of p38alpha MAPK by non-radioactive immunosorbent assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50243761(4-(1H-Indol-3-yl)-3-(3,4,5-trimethoxyphenyl)-1,5-d...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FQSPubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen

Curated by ChEMBL
LigandPNGBDBM50516609(CHEMBL4445595)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2ZWXPubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50243761(4-(1H-Indol-3-yl)-3-(3,4,5-trimethoxyphenyl)-1,5-d...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FQSPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of rat recombinant GST-tagged CK1delta using GST-tagged mouse p53 (1 to 64 residues) as substrate in presence of radiolabelled-ATP by Cher...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50428028(CHEMBL1257064)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of rat GST-tagged CK1delta M82F mutant at 10 uM using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50025020(CHEMBL3337854)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of human CK1delta transcription variant 2 using GST-tagged mouse p53 (1 to 64 residues) as substrate in presence of radiolabelled-ATP by C...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM13531(4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridy...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50455468(CHEMBL1257114)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of rat GST-tagged CK1delta M82F mutant at 10 uM using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4F5DPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300886(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)-N-...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50182470(5,6,7-trimethoxy-1,2,3,8-tetrahydro-benzo[a]pyrrol...)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of human VEGFR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC108SPubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant CK1epsilon by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50455466(CHEMBL4204681)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of rat recombinant CK1delta kinase domain using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4F5DPubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50455466(CHEMBL4204681)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of rat GST-tagged CK1delta M82F mutant at 10 uM using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4F5DPubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen

Curated by ChEMBL
LigandPNGBDBM50516607(CHEMBL4530882)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2ZWXPubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Christian-Albrechts-University of Kiel

Curated by ChEMBL
LigandPNGBDBM50192871(CHEMBL3358996)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant PDGFRbeta using poly(Ala,Glu,Lys,Tyr) substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZG6V0RPubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen

Curated by ChEMBL
LigandPNGBDBM50516620(CHEMBL4557039)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2ZWXPubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K7961PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50588635(CHEMBL5186013)copy SMILES
Affinity DataIC50: 120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7FFTPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50004566(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinaz...)copy SMILEScopy InChI
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7FFTPubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50428027(CHEMBL1257090)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of rat GST-tagged CK1delta M82F mutant at 10 uM using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4F5DPubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls-University

Curated by ChEMBL
LigandPNGBDBM50365355(CHEMBL1257089)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of rat GST-tagged CK1delta M82F mutant at 10 uM using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4F5DPubMed
TargetProtein-serine O-palmitoleoyltransferase porcupine(Homo sapiens (Human))
Ulm University Hospital

Curated by ChEMBL
LigandPNGBDBM50428028(CHEMBL1257064)copy SMILEScopy InChI
Affinity DataIC50: 157nMAssay Description:Inhibition of porcupine in HEK293T cells transfected with Wnt3A-expressing vector assessed as suppression of Wnt/beta-catenin signaling after 22 hrs ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4F5DPubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Medical Center Groningen

Curated by ChEMBL
LigandPNGBDBM50516612(CHEMBL4527473)copy SMILEScopy InChI
Affinity DataIC50: 157nMAssay Description:Inhibition of human recombinant N-terminal GST/His6-tagged BRAF V600E mutant (Q417 to H766 residues) expressed in Sf9 insect cells using MEK1 as subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2ZWXPubMed
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