Compile Data Set for Download or QSAR
Found 49 with Last Name = 'pouget' and Initial = 'c'
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMedDrugBank
TargetAromatase [1-48](Homo sapiens (Human))
Biomolécules et Cibles Cellulaires Tumorales

LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6P2ZPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345191(7,8-Benzo-4'-hydroxy-4-imidazolylflavan | CHEMBL17...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345189(2,4-trans-7,8-benzo-4-imidazolylflavan | CHEMBL178...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50118965(4-Imidazol-1-yl-2-phenyl-chroman-7-ol | CHEMBL9591...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1WQ8PubMed
TargetAromatase [1-48](Homo sapiens (Human))
Biomolécules et Cibles Cellulaires Tumorales

LigandPNGBDBM85252(2,4-Trans-4'-hydroxy-4-imidazolyl-7-methoxyfla...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6P2ZPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50118965(4-Imidazol-1-yl-2-phenyl-chroman-7-ol | CHEMBL9591...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PK0FHSPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase [1-48](Homo sapiens (Human))
Biomolécules et Cibles Cellulaires Tumorales

LigandPNGBDBM85253(2,4-Trans-4',7-dihydroxy-4-imidazolyl-7-methox...)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6P2ZPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1WQ8PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PK0FHSPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase [1-48](Homo sapiens (Human))
Biomolécules et Cibles Cellulaires Tumorales

LigandPNGBDBM85249(2,4-Trans-3'-hydroxy-4-imidazolyl-7-methoxyfla...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6P2ZPubMed
TargetAromatase [1-48](Homo sapiens (Human))
Biomolécules et Cibles Cellulaires Tumorales

LigandPNGBDBM85251(2,4-Trans-4'-cyano-4-imidazolyl-7-methoxyflava...)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6P2ZPubMed
TargetAromatase [1-48](Homo sapiens (Human))
Biomolécules et Cibles Cellulaires Tumorales

LigandPNGBDBM85250(2,4-Trans-4'-chloro-4-imidazolyl-7-methoxyflav...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6P2ZPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50153525(2-Phenyl-4-[1,2,4]triazol-1-yl-chroman-7-ol | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1WQ8PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)copy SMILEScopy InChI
Affinity DataIC50: 534nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)copy SMILEScopy InChI
Affinity DataIC50: 534nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50374254(CHEMBL439241)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50111269(7-Methoxy-2-phenyl-3-pyridin-4-ylmethylene-chroman...)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125S01PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345188(2-(4-hydroxyphenyl)-2,3-dihydrobenzo[h]chromen-4-o...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345188(2-(4-hydroxyphenyl)-2,3-dihydrobenzo[h]chromen-4-o...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50111268(2-Phenyl-3-pyridin-4-ylmethylene-chroman-4-one | C...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125S01PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50374255(CHEMBL258257)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50153523(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-[1,2,4]tria...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1WQ8PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345187(4-(4-oxo-3,4-dihydro-2H-benzo[h]chromen-2-yl)benzo...)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345187(4-(4-oxo-3,4-dihydro-2H-benzo[h]chromen-2-yl)benzo...)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50111270(7-Methoxy-2-phenyl-3-pyridin-4-ylmethylene-chroman...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125S01PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50014323(2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50241408((2S)-liquiritigenin | 7-HYDROXY-2-(4-HYDROXY-PHENY...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50111271(2-Phenyl-3-pyridin-4-ylmethylene-chroman-4-one | C...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125S01PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50374256(CHEMBL255110)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50374258(CHEMBL256407)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50374257(CHEMBL402970)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50104887(2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PK0FHSPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50104887(2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345186(2-phenyl-2,3-dihydrobenzo[h]chromen-4-one | 2-phen...)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50345186(2-phenyl-2,3-dihydrobenzo[h]chromen-4-one | 2-phen...)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)copy SMILEScopy InChI
Affinity DataIC50: 5.20E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125S01PubMedDrugBank
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)copy SMILEScopy InChI
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PK0FHSPubMedDrugBank
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC90CBPubMedDrugBank
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50106920((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50106920((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PK0FHSPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50106920((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125S01PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50051358(2,3-Dihydroflavone | 2,3-dihydro-2-phenyl-4H-1-ben...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DR2WCCPubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50051358(2,3-Dihydroflavone | 2,3-dihydro-2-phenyl-4H-1-ben...)copy SMILEScopy InChI
Affinity DataIC50: 2.85E+4nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125S01PubMed
TargetAromatase(Homo sapiens (Human))
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales

Curated by ChEMBL
LigandPNGBDBM50153524(4-(7-Methoxy-2-phenyl-chroman-4-yl)-4H-[1,2,4]tria...)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1WQ8PubMed