TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
TargetGlucagon receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH and Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH and Co. KG
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human PPARgamma receptor assessed as rosiglitazone-induced receptor activation by alphascreen assayMore data for this Ligand-Target Pair
TargetGlucagon receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH and Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH and Co. KG
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of His-tagged human src kinase expressed in Sf9 cells by DELFIA assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at human PPARgamma receptor in CHO-K1 cells assessed as rosiglitazone-induced receptor activation by cell based reporter assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of His-tagged human src kinase expressed in Sf9 cells by DELFIA assayMore data for this Ligand-Target Pair
TargetGlucagon receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH and Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH and Co. KG
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human glucagon receptor expressed in BHK21 cells assessed as inhibition of glucagon-induced cAMP elevation by RIAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of His-tagged human src kinase expressed in Sf9 cells by DELFIA assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 3.75E+4nMAssay Description:Inhibition of His-tagged human src kinase expressed in Sf9 cells by DELFIA assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of His-tagged human src kinase expressed in Sf9 cells by DELFIA assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Boehringer Ingelheim Pharma GmbH & Co. KG
Curated by ChEMBL
Affinity DataEC50: 260nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
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