Compile Data Set for Download or QSAR
Found 269 with Last Name = 'sargent' and Initial = 'c'
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344999(2-(2'-chloro-4'-(N-methylmethylsulfonamido)-5-(tri...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344993(2-(2'-chloro-4'-(methylsulfonyl)-5-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344995(2-(5'-cyano-2'-methyl-5-(trifluoromethyl)biphenyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344996(2-(5'-cyano-2'-fluoro-5-(trifluoromethyl)biphenyl-...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339747((S)-2-(2-((4-(2-(4-fluorophenyl)acetyl)-3-methylpi...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344992(2-(2'-chloro-4'-(ethylsulfonyl)-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344998(2-(2'-methyl-4'-(N-methylmethylsulfonamido)-5-(tri...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50026419(CHEMBL1778628)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339748(CHEMBL1689128 | [4-Chloro-2-[[(3S)-4-[(4-chlorophe...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344988(2-(2',5-dichloro-4'-(methylsulfonyl)biphenyl-2-ylo...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344975((2R)-2-(2'-chloro-4'-(ethylsulfonyl)-5-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344974((R)-2-(3'-cyano-5-(trifluoromethyl)biphenyl-2-ylox...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339749((S)-2-(2-((4-(benzylsulfonyl)-3-methylpiperazin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357127(CHEMBL1917440)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50345003(2-(4'-(N-methylmethylsulfonamido)-5-(trifluorometh...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339750((S)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)pip...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344991(2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357125(CHEMBL1917438)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339751((S)-2-(4-chloro-2-((4-(2-(4-fluorophenyl)acetyl)-3...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Mus musculus (mouse))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344991(2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Binding affinity to mouse CRTh2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339752((S)-2-(4-chloro-2-((4-(phenylsulfonyl)-3-propylpip...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Rattus norvegicus)
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344991(2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Binding affinity to rat CRTh2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357112(CHEMBL1917427)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339753((S)-2-(4-chloro-2-(((S)-4-(2-(4-chlorophenyl)acety...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50345007(2-(4'-(N,N-diethylsulfamoyl)-5-(trifluoromethyl)bi...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357105(CHEMBL1917443)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344984(2-(2',5-dichloro-4'-(ethylsulfonyl)biphenyl-2-ylox...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344982((2R)-2-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357149(CHEMBL1917426)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344994(2-(5-chloro-3'-cyanobiphenyl-2-yloxy)acetic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357104(CHEMBL1917433)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50345001((5-Trifluoromethyl-[1,1':2',1'']terphenyl-2-yloxy)...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339754(CHEMBL1689135 | [4-Chloro-2-({(3S)-4-[(4-chlorophe...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344997(2-(2'-chloro-5-fluoro-4'-(N-methylmethylsulfonamid...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344978(3-(4'-(ethylsulfonyl)-2'-methyl-5-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357129(CHEMBL1917442)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357128(CHEMBL1917441)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339755((S)-2-(4-chloro-2-((3-methyl-4-(2-phenylacetyl)pip...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357144(CHEMBL1917458)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357142(CHEMBL1917456)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357124(CHEMBL1917437)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357126(CHEMBL1917439)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357146(CHEMBL1917460)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50344985(2-(5-chloro-4'-(ethylsulfonyl)-2'-methylbiphenyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Displacement of [3H]-PGD2 from CRTh2 receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46S9ZPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357102(CHEMBL1914489)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339750((S)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)pip...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50339756((S)-2-(4-chloro-2-((3-ethyl-4-(phenylsulfonyl)pipe...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41RQJPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085853(CHEMBL173251 | Sodium; [2-cyano-5-(pyridin-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065508((R)-4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM594WPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
AstraZeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50357140(CHEMBL1917454)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3225PubMed
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