Compile Data Set for Download or QSAR
Found 134 with Last Name = 'spanier' and Initial = 'c'
TargetP2X purinoceptor 1(RAT)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50240455(CHEMBL1253351)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Antagonist activity at rat P2X1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(RAT)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540410(CHEMBL337395)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Antagonist activity at rat P2X1 receptorMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430160(CHEMBL536151 | TCMDC-125465)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430195(CHEMBL2338696)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430185(CHEMBL2179173)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540434(CHEMBL4640175)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430177(CHEMBL2088014)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540434(CHEMBL4640175)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430156(CHEMBL2338695)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540436(CHEMBL2179174)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430156(CHEMBL2338695)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430185(CHEMBL2179173)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540422(CHEMBL4644398)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540442(CHEMBL2088011)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430159(CHEMBL461542)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430176(CHEMBL589733 | MMV665807 | SJ000010289)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540442(CHEMBL2088011)copy SMILEScopy InChI
Affinity DataIC50: 135nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540434(CHEMBL4640175)copy SMILEScopy InChI
Affinity DataIC50: 143nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430159(CHEMBL461542)copy SMILEScopy InChI
Affinity DataIC50: 155nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540436(CHEMBL2179174)copy SMILEScopy InChI
Affinity DataIC50: 155nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430160(CHEMBL536151 | TCMDC-125465)copy SMILEScopy InChI
Affinity DataIC50: 156nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540436(CHEMBL2179174)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540439(CHEMBL2088009)copy SMILEScopy InChI
Affinity DataIC50: 172nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430160(CHEMBL536151 | TCMDC-125465)copy SMILEScopy InChI
Affinity DataIC50: 175nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430156(CHEMBL2338695)copy SMILEScopy InChI
Affinity DataIC50: 177nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430170(CHEMBL2338686)copy SMILEScopy InChI
Affinity DataIC50: 195nMAssay Description:Antagonist activity at human P2X3 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430195(CHEMBL2338696)copy SMILEScopy InChI
Affinity DataIC50: 196nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540432(CHEMBL2088012)copy SMILEScopy InChI
Affinity DataIC50: 199nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430195(CHEMBL2338696)copy SMILEScopy InChI
Affinity DataIC50: 209nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540449(CHEMBL4637528)copy SMILEScopy InChI
Affinity DataIC50: 219nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430194(CHEMBL2313115)copy SMILEScopy InChI
Affinity DataIC50: 236nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50240455(CHEMBL1253351)copy SMILEScopy InChI
Affinity DataIC50: 236nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430159(CHEMBL461542)copy SMILEScopy InChI
Affinity DataIC50: 315nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430186(CHEMBL2178702)copy SMILEScopy InChI
Affinity DataIC50: 323nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540443(CHEMBL4648128)copy SMILEScopy InChI
Affinity DataIC50: 335nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430170(CHEMBL2338686)copy SMILEScopy InChI
Affinity DataIC50: 341nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430177(CHEMBL2088014)copy SMILEScopy InChI
Affinity DataIC50: 371nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540456(CHEMBL2313133)copy SMILEScopy InChI
Affinity DataIC50: 439nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50168286(1H-Benzoimidazole-2-carboxylic acid [(R)-1-((1S,2R...)copy SMILEScopy InChI
Affinity DataIC50: 496nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540441(CHEMBL2179168)copy SMILEScopy InChI
Affinity DataIC50: 522nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430176(CHEMBL589733 | MMV665807 | SJ000010289)copy SMILEScopy InChI
Affinity DataIC50: 537nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540444(CHEMBL2179170)copy SMILEScopy InChI
Affinity DataIC50: 567nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430160(CHEMBL536151 | TCMDC-125465)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Antagonist activity P2X1 receptor in Apyrase pre-treated human platelets assessed as inhibition of collagen-induced platelet aggregation pre-incubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540442(CHEMBL2088011)copy SMILEScopy InChI
Affinity DataIC50: 599nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540423(CHEMBL4639803)copy SMILEScopy InChI
Affinity DataIC50: 655nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430185(CHEMBL2179173)copy SMILEScopy InChI
Affinity DataIC50: 712nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430170(CHEMBL2338686)copy SMILEScopy InChI
Affinity DataIC50: 729nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430193(CHEMBL2313119)copy SMILEScopy InChI
Affinity DataIC50: 755nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50430170(CHEMBL2338686)copy SMILEScopy InChI
Affinity DataIC50: 797nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50540422(CHEMBL4644398)copy SMILEScopy InChI
Affinity DataIC50: 857nMAssay Description:Antagonist activity at human P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V93PubMed
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