Compile Data Set for Download or QSAR
Found 41 with Last Name = 'spickler' and Initial = 'c'
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005004(CHEMBL2397309)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005008(CHEMBL2397312)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005009(CHEMBL2397311)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436476(CHEMBL2397316)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005007(CHEMBL2397310)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005010(CHEMBL2397313)copy SMILEScopy InChI
Affinity DataIC50: 67nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005011(CHEMBL2397303)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005005(CHEMBL2397317)copy SMILEScopy InChI
Affinity DataIC50: 137nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-kinase beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436478(CHEMBL2397314)copy SMILEScopy InChI
Affinity DataIC50: 225nMAssay Description:Inhibition of PI4K3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005011(CHEMBL2397303)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436481(CHEMBL2397305)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005006(CHEMBL2397307)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436482(CHEMBL2397304)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436476(CHEMBL2397316)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of STK17A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436482(CHEMBL2397304)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436478(CHEMBL2397314)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of STK17A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436481(CHEMBL2397305)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetRibosomal protein S6 kinase alpha-4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436476(CHEMBL2397316)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of MSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PIK3C2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436476(CHEMBL2397316)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of PIK3C2B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005010(CHEMBL2397313)copy SMILEScopy InChI
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of MAP4K4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of PIK3C2B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436478(CHEMBL2397314)copy SMILEScopy InChI
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of MAP4K2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DYRK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of PIK3CD (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetPhosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436476(CHEMBL2397316)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of PIK3C2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436479(CHEMBL2397308)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436476(CHEMBL2397316)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005009(CHEMBL2397311)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436480(CHEMBL2397306)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005008(CHEMBL2397312)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436477(CHEMBL2397315)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436480(CHEMBL2397306)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436479(CHEMBL2397308)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005005(CHEMBL2397317)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005007(CHEMBL2397310)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50436478(CHEMBL2397314)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Boehringer Ingelheim (Canada) Ltd.

Curated by ChEMBL
LigandPNGBDBM50005004(CHEMBL2397309)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2QCXPubMed