Compile Data Set for Download or QSAR
Found 333 with Last Name = 'strathdee' and Initial = 'c'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400752(CHEMBL2203552)copy SMILEScopy InChI
Affinity DataIC50: 1.49nMAssay Description:Inhibition of GSK3betaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400756(CHEMBL2203562)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400754(CHEMBL2203564)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetG protein-coupled receptor kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50566950(CHEMBL4852125)copy SMILES
Affinity DataIC50: 3.5nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetG protein-coupled receptor kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50566949(CHEMBL4877302)copy SMILES
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human GRK6 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400753(CHEMBL2203565)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400757(CHEMBL2203561)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400755(CHEMBL2203563)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
TargetG protein-coupled receptor kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50566953(CHEMBL4860332)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetRhodopsin kinase GRK7(Homo sapiens (Human))TBA
LigandPNGBDBM50566949(CHEMBL4877302)copy SMILES
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant full length human GRK7 using casein as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetG protein-coupled receptor kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50566946(CHEMBL4854871)copy SMILES
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetG protein-coupled receptor kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50566949(CHEMBL4877302)copy SMILES
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400748(CHEMBL2203556)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400752(CHEMBL2203552)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400752(CHEMBL2203552)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of CK1-alpha using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 8 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetG protein-coupled receptor kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50566923(CHEMBL4855000)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50566915(CHEMBL4848826)copy SMILES
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant full length human Aurora A using LRRASLG as substrate incubated for 40 mins in presence of [gamma-33ATP] by radiometric sci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetG protein-coupled receptor kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM50566951(CHEMBL4875929)copy SMILES
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))TBA
LigandPNGBDBM50566949(CHEMBL4877302)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant full length human GRK5 using casein as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
TargetRhodopsin kinase GRK7(Homo sapiens (Human))TBA
LigandPNGBDBM50566946(CHEMBL4854871)copy SMILES
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant full length human GRK7 using casein as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2D97PubMed
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