Compile Data Set for Download or QSAR
Found 193 with Last Name = 'tahtaoui' and Initial = 'c'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151212(CHEMBL2368393 | difluoro(2-{[(2Z)-1-methyl-5-[2-({...)copy SMILEScopy InChI
Affinity DataKi:  8.80nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151218(CHEMBL2368392 | difluoro(2-{[(2Z)-1-methyl-5-(2-{[...)copy SMILEScopy InChI
Affinity DataKi:  8.90nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)copy SMILEScopy InChI
Affinity DataKi:  23.5nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16GNPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50178133(1-ethyl-2-[(1E,3E)-3-(1-ethylquinolin-2-(1H)-ylide...)copy SMILEScopy InChI
Affinity DataKi:  29.4nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16GNPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151214(CHEMBL2368390 | difluoro(2-{[(2Z)-1-methyl-5-[2-({...)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50178130(CHEMBL220095 | RR(17)PZ)copy SMILEScopy InChI
Affinity DataKi:  53.5nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16GNPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151215(2-[6-(diethylamino)-3-(diethyliminiumyl)-3H-xanthe...)copy SMILEScopy InChI
Affinity DataKi:  54nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151216(CHEMBL2368391 | difluoro(2-{[(2Z)-1-methyl-5-{2-[(...)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50178128(Bo(15)PZ | CHEMBL198982)copy SMILEScopy InChI
Affinity DataKi:  69.7nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16GNPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151213(CHEMBL365702 | difluoro(2-{[(2Z)-1-methyl-5-(2-{[5...)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151219((2E)-2-[(2E)-3-[3,3-dimethyl-1-(5-{[2-(2-{2-[4-(2-...)copy SMILEScopy InChI
Affinity DataKi:  135nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50178129(2-{[4-(diethylamino)phenyl][4-(diethyliminio)cyclo...)copy SMILEScopy InChI
Affinity DataKi:  189nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16GNPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151211(2,2-difluoro-12-[2-(methylcarbamoyl)ethyl]-4-(thio...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50151217(CHEMBL2368394 | difluoro(2-{[(2Z)-1-methyl-5-[2-({...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43TVQPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50178131(6-[(5-carboxypentanoyl)amino]-1-ethyl-2-[(1E,3E)-3...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16GNPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
UMR CNRS/ULP 7081

Curated by ChEMBL
LigandPNGBDBM50178132(CHEMBL370564 | {4-[[4-(5-carboxy-pentylsulfamoyl)-...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]QNB from EGFP(delta17)human M1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB16GNPubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270876(US10059709, 22)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410174(US10370375, Example 22)copy SMILES
Affinity DataIC50: 10nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410170(US10370375, Example 18)copy SMILES
Affinity DataIC50: 21nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270872(US10059709, 18)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270880(US10059709, 26)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410178(US10370375, Example 26)copy SMILES
Affinity DataIC50: 34nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270879(US10059709, 25)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410177(US10370375, Example 25)copy SMILES
Affinity DataIC50: 71nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270876(US10059709, 22)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2 [888-1187](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410174(US10370375, Example 22)copy SMILES
Affinity DataIC50: 130nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK3 [811-1124](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410174(US10370375, Example 22)copy SMILES
Affinity DataIC50: 260nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270876(US10059709, 22)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270872(US10059709, 18)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2 [888-1187](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410170(US10370375, Example 18)copy SMILES
Affinity DataIC50: 390nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410180(US10370375, Example 28)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270882(US10059709, 28)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270856(US10059709, 2)copy SMILEScopy InChI
Affinity DataIC50: 582nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410154(US10370375, Example 2)copy SMILES
Affinity DataIC50: 582nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270855(US10059709, 1)copy SMILEScopy InChI
Affinity DataIC50: 838nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410153(US10370375, Example 1)copy SMILES
Affinity DataIC50: 838nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270880(US10059709, 26)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2 [888-1187](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410178(US10370375, Example 26)copy SMILES
Affinity DataIC50: 840nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270878(US10059709, 24)copy SMILEScopy InChI
Affinity DataIC50: 930nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410176(US10370375, Example 24)copy SMILEScopy InChI
Affinity DataIC50: 930nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270879(US10059709, 25)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetNon-receptor tyrosine-protein kinase TYK2 [888-1187](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410177(US10370375, Example 25)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK3 [811-1124](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410170(US10370375, Example 18)copy SMILES
Affinity DataIC50: 1.20E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270872(US10059709, 18)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270881(US10059709, 27)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410179(US10370375, Example 27)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM270856(US10059709, 2)copy SMILEScopy InChI
Affinity DataIC50: 1.89E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25X2BZXUS Patent
TargetTyrosine-protein kinase JAK3 [811-1124](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410154(US10370375, Example 2)copy SMILES
Affinity DataIC50: 1.89E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
TargetTyrosine-protein kinase JAK1 [866-1154](Homo sapiens (Human))
Elanco Tiergesundheit AG

US Patent
LigandPNGBDBM410165(US10370375, Example 13)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:All four kinases of the JAK/TYK-kinase family were used as purified recombinant GST-fusion proteins, containing the active kinase domains. GST-JAK1(8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC857BUS Patent
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