TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (electrogenicity) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataKi: 5.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.1 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the presence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the absence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the presence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the presence of bicarbonate) (TEA: 20 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the absence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the absence of bicarbonate) (TEA: 20 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 2.56E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant SIRT3 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the presence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 7.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.13E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the absence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.27E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the presence of bicarbonate) (TEA: 20 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.46E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of Amantadine uptake (in the presence of bicarbonate) (Amantadine: 10 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 1.75E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(Homo sapiens (Human))
Institut f£r Physiologie
Curated by ChEMBL
Institut f£r Physiologie
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of Dopamine uptake (Dopamine: 200 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 3.70E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 2(RAT)
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Institute of Anatomy of the Bayerische Julius-Maximilians-Universit£t
Curated by ChEMBL
Affinity DataIC50: 3.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the absence of bicarbonate) (TEA: 20 uM) in OCT2-expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT3 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT1 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT1 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT1 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT1 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT3 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT3 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT3 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT3 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT3 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT1 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT1 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant SIRT2 using fluorescent peptide substrate by fluorescent assayMore data for this Ligand-Target Pair