Compile Data Set for Download or QSAR
Found 37 with Last Name = 'westerlund' and Initial = 'c'
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228308(CHEMBL413740)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228272(CHEMBL411997)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50471553(CHEMBL1791261)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228195(Angiotensin Ii | CHEBI:2719)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228272(CHEMBL411997)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat uterine membranes (Angiotensin II receptor, type 1)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228308(CHEMBL413740)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat uterine membranes (Angiotensin II receptor, type 1)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50471554(CHEMBL1791267)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228196(CHEMBL405464)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228308(CHEMBL413740)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat pituitary membranes (Angiotensin II receptor, type 1) in presence of 0.2% b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228272(CHEMBL411997)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat pituitary membranes (Angiotensin II receptor, type 1) in presence of 0.2% b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228196(CHEMBL405464)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat pituitary membranes (Angiotensin II receptor, type 1) in presence of 0.2% b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50228196(CHEMBL405464)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibitory concentration against specific binding of [125 I]Ang II to rat uterine membranes (Angiotensin II receptor, type 1)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402953(CHEMBL2206790)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402952(CHEMBL2206791)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402951(CHEMBL2206792)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50471552(CHEMBL1791262)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50369331(CHEMBL1791259)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against [125 I]Ang II binding to rat pituitary membranes Angiotensin II receptor type 1 without 0.2% bovine serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4SM4PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402962(CHEMBL2206778)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402963(CHEMBL2206777)copy SMILEScopy InChI
Affinity DataEC50:  501nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402964(CHEMBL2206776)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402965(CHEMBL1401244)copy SMILEScopy InChI
Affinity DataEC50:  2.51E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402958(CHEMBL2206782)copy SMILEScopy InChI
Affinity DataEC50:  3.16E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402957(CHEMBL2206783)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402956(CHEMBL2206784)copy SMILEScopy InChI
Affinity DataEC50:  1.58E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402955(CHEMBL2206785)copy SMILEScopy InChI
Affinity DataEC50:  126nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402953(CHEMBL2206790)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402954(CHEMBL2206787)copy SMILEScopy InChI
Affinity DataEC50:  316nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402952(CHEMBL2206791)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402951(CHEMBL2206792)copy SMILEScopy InChI
Affinity DataEC50:  200nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402953(CHEMBL2206790)copy SMILEScopy InChI
Affinity DataEC50:  50.1nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402952(CHEMBL2206791)copy SMILEScopy InChI
Affinity DataEC50:  63.1nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402951(CHEMBL2206792)copy SMILEScopy InChI
Affinity DataEC50:  126nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402950(CHEMBL2206775)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402959(CHEMBL2206781)copy SMILEScopy InChI
Affinity DataEC50:  794nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402960(CHEMBL2206780)copy SMILEScopy InChI
Affinity DataEC50:  631nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed
TargetHexokinase-4(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50402961(CHEMBL2206779)copy SMILEScopy InChI
Affinity DataEC50:  1.58E+4nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BK1DJ3PubMed